SCHEMBL7723247

SCHEMBL7723247

Cc1cc2nc(C(O)[C@@H](CCc3ccccc3)N(C(=O)OC(C)(C)C)C(=O)[C@H](N)CCCNC(=O)OC(C)(C)C)oc2cc1C

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 2/20 0.38
NPSR1 Q6W5P4 2/20 0.36
MMP1 P03956 1/20 0.35
MMP3 P08254 1/20 0.35
MMP9 P14780 1/20 0.35
CTSK P43235 2/20 0.35
BRD4 O60885 6/20 0.34
ATM Q13315 1/20 0.34
SIGMAR1 Q99720 2/20 0.34
CTSS P25774 1/20 0.33
JAK2 O60674 1/20 0.33
S1PR4 O95977 1/20 0.33
ALDH1A1 P00352 1/20 0.33
LMNA P02545 1/20 0.33
HSP90AA1 P07900 1/20 0.33
THRB P10828 1/20 0.33
HPGD P15428 1/20 0.33
XBP1 P17861 1/20 0.33
HTT P42858 1/20 0.33
POLB P06746 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7731104 0.91 MAPT (0.39) MAPTNPSR1MMP1MMP3MMP9
SCHEMBL7731051 0.90 LMNA (0.39) MAPTNPSR1MMP1MMP3MMP9
SCHEMBL7735575 0.90 MAPT (0.37) MAPTNPSR1MMP1MMP3MMP9
SCHEMBL7723226 0.86 MAPT (0.38) MAPTNPSR1MMP1MMP3MMP9
SCHEMBL7732168 0.80 ADORA3 (0.37) MAPTNPSR1MMP1MMP3MMP9
SCHEMBL7731071 0.79 BCHE (0.45) NPSR1MMP1MMP3MMP9CTSK
SCHEMBL7731093 0.79 MAPT (0.41) MAPTNPSR1MMP1MMP3MMP9
SCHEMBL7730530 0.72 MAPT (0.38) MAPTNPSR1MMP1MMP3MMP9
SCHEMBL7723327 0.72 MAPT (0.44) MAPTNPSR1MMP1MMP3MMP9
SCHEMBL7730106 0.70 CTSC (0.38) CTSKCTSS

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6436980-B1 TRANSPORT PROTEIN SUPPRESSORS; MICROBIOCIDES ESSENTIAL THERAPEUTICS, INC. 2002-08-20 US disclosed
US-6204279-B1 SECONDARY AMIDE CONTAINING BENZOXAZOLE DERIVATIVES MICROCIDE PHARMACEUTICALS, INC. 2001-03-20 US disclosed