SCHEMBL7731093

SCHEMBL7731093

Cc1cc2nc(C(O)[C@@H](CCc3ccccc3)NCC(O)[C@@H](CCCNC(=O)OC(C)(C)C)NC(=O)OC(C)(C)C)oc2cc1C

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 2/20 0.41
NPSR1 Q6W5P4 2/20 0.38
CTSK P43235 3/20 0.37
CTSS P25774 1/20 0.37
MMP1 P03956 1/20 0.37
MMP3 P08254 1/20 0.37
MMP9 P14780 1/20 0.37
ATM Q13315 1/20 0.36
KLK5 Q9Y337 1/20 0.35
ALDH1A1 P00352 3/20 0.35
LMNA P02545 2/20 0.35
BRD4 O60885 2/20 0.35
POLB P06746 1/20 0.35
JAK2 O60674 1/20 0.35
S1PR4 O95977 1/20 0.35
HSP90AA1 P07900 1/20 0.35
THRB P10828 1/20 0.35
HPGD P15428 1/20 0.35
XBP1 P17861 1/20 0.35
HTT P42858 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7723247 0.79 MAPT (0.38) MAPTNPSR1CTSKCTSSMMP1
SCHEMBL5731227 0.77 CTSK (0.46) MAPTNPSR1CTSKCTSSATM
SCHEMBL5731226 0.77 CTSK (0.46) MAPTNPSR1CTSKCTSSATM
SCHEMBL7734143 0.76 ATM (0.46) ATM
Trifluoroacetic Acid SCHEMBL7735796 0.75 HRH2 (0.34) MAPT
SCHEMBL12247706 0.73 MAPT (0.59) MAPTNPSR1KLK5POLBMEN1
SCHEMBL7730106 0.72 CTSC (0.38) CTSKCTSS
SCHEMBL7735797 0.71 METAP2 (0.32)
SCHEMBL7731132 0.70 HDAC4 (0.43) MAPTNPSR1MMP1MMP3MMP9
Trifluoroacetic Acid SCHEMBL7734181 0.70 OPRK1 (0.37)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6436980-B1 TRANSPORT PROTEIN SUPPRESSORS; MICROBIOCIDES ESSENTIAL THERAPEUTICS, INC. 2002-08-20 US disclosed