SCHEMBL7723640

SCHEMBL7723640

CCOC(=O)Cn1nc(-c2ccc(OC)cc2)cc(C(=O)NC)c1=O

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.52
KDM4E B2RXH2 3/20 0.52
SMN1; SMN2 Q16637 2/20 0.52
HSD17B10 Q99714 1/20 0.52
KMT2A Q03164 3/20 0.52
MEN1 O00255 1/20 0.52
TSHR P16473 2/20 0.50
MAPK1 P28482 1/20 0.49
HTT P42858 2/20 0.49
MAPT P10636 1/20 0.48
TDP1 Q9NUW8 2/20 0.46
GLA P06280 1/20 0.46
HPGD P15428 1/20 0.46
UBE2N P61088 1/20 0.46
NPC1 O15118 1/20 0.45
LMNA P02545 2/20 0.45
POLB P06746 2/20 0.45
JAK2 O60674 1/20 0.45
PKM P14618 1/20 0.44
APEX1 P27695 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7723506 0.88 MAPT (0.55) ALDH1A1KDM4ESMN1; SMN2HSD17B10KMT2A
SCHEMBL7730172 0.87 LMNA (0.51) ALDH1A1KDM4EKMT2AMEN1MAPT
SCHEMBL7725155 0.87 JAK2 (0.47) ALDH1A1KDM4EKMT2AHTTMAPT
SCHEMBL7724719 0.85 JAK2 (0.45) ALDH1A1KDM4ESMN1; SMN2HSD17B10KMT2A
SCHEMBL7726296 0.83 JAK2 (0.45) ALDH1A1KDM4EHSD17B10KMT2AMEN1
SCHEMBL7720154 0.82 JAK2 (0.44) ALDH1A1KDM4EKMT2AHTTMAPT
SCHEMBL7724650 0.82 RAB9A (0.49) ALDH1A1KDM4EHSD17B10KMT2AMAPT
SCHEMBL7720252 0.81 ALDH1A1 (0.47) ALDH1A1KDM4EKMT2AHTTMAPT
SCHEMBL7723523 0.80 CRHR1 (0.51) ALDH1A1KDM4EHTTNPC1LMNA
SCHEMBL7720270 0.80 MAPT (0.59) ALDH1A1SMN1; SMN2KMT2AMEN1HTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6403586-B1 Pyridazine derivatives and drugs containing the same as the active ingredient KOWA CO., LTD. (JP) 2002-06-11 US disclosed
EP-1061077-A1 NOVEL PYRIDAZINE DERIVATIVES AND DRUGS CONTAINING THE SAME AS THE ACTIVE INGREDIENT Kowa Co., Ltd. (JP) 2000-12-20 EP disclosed