SCHEMBL7730172

SCHEMBL7730172

CNC(=O)Cn1nc(-c2ccc(OC)cc2)cc(C(=O)NC)c1=O

nearest known ligand 0.52

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
LMNA P02545 2/20 0.51
KMT2A Q03164 3/20 0.49
MAPT P10636 2/20 0.48
JAK2 O60674 1/20 0.47
MEN1 O00255 1/20 0.47
RXFP1 Q9HBX9 1/20 0.47
ALDH1A1 P00352 2/20 0.47
RECQL P46063 1/20 0.47
POLB P06746 1/20 0.47
TDP1 Q9NUW8 1/20 0.46
CACNA1B Q00975 1/20 0.46
APBA1 Q02410 1/20 0.46
FPR1 P21462 1/20 0.45
FPR2 P25090 1/20 0.45
RAB9A P51151 1/20 0.45
KDM4E B2RXH2 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7724650 0.90 RAB9A (0.49) LMNAKMT2AMAPTALDH1A1POLB
SCHEMBL7725155 0.88 JAK2 (0.47) LMNAKMT2AMAPTJAK2ALDH1A1
SCHEMBL7723640 0.87 ALDH1A1 (0.52) LMNAKMT2AMAPTJAK2MEN1
SCHEMBL7726296 0.86 JAK2 (0.45) LMNAKMT2AMAPTJAK2MEN1
SCHEMBL7724719 0.86 JAK2 (0.45) LMNAKMT2AMAPTJAK2ALDH1A1
SCHEMBL7720154 0.85 JAK2 (0.44) LMNAKMT2AMAPTJAK2ALDH1A1
SCHEMBL7726424 0.85 KMT2A (0.54) LMNAKMT2AMAPTMEN1RXFP1
SCHEMBL7720252 0.84 ALDH1A1 (0.47) LMNAKMT2AMAPTJAK2ALDH1A1
SCHEMBL7730164 0.84 ADORA2A (0.54) KMT2AMAPTMEN1RXFP1ALDH1A1
SCHEMBL7723582 0.84 ALDH1A1 (0.44) LMNAKMT2AMAPTJAK2ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6403586-B1 Pyridazine derivatives and drugs containing the same as the active ingredient KOWA CO., LTD. (JP) 2002-06-11 US disclosed
EP-1061077-A1 NOVEL PYRIDAZINE DERIVATIVES AND DRUGS CONTAINING THE SAME AS THE ACTIVE INGREDIENT Kowa Co., Ltd. (JP) 2000-12-20 EP disclosed