SCHEMBL7730177

SCHEMBL7730177

CCOC(=O)Nc1cc(-c2ccc(OC)cc2)nn(CC2CC2)c1=O

nearest known ligand 0.49

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
L3MBTL1 Q9Y468 1/20 0.49
LMNA P02545 2/20 0.48
CRHR1 P34998 1/20 0.47
MAPT P10636 1/20 0.46
POLB P06746 2/20 0.45
FAAH O00519 2/20 0.45
ALDH1A1 P00352 2/20 0.45
KDM4E B2RXH2 1/20 0.44
RAB9A P51151 1/20 0.44
CTSL P07711 1/20 0.42
CTSB P07858 1/20 0.42
PTGIR P43119 1/20 0.41
RECQL P46063 1/20 0.41
KMT2A Q03164 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7724779 0.84 MAPT (0.53) L3MBTL1LMNACRHR1MAPTPOLB
SCHEMBL7724785 0.83 LMNA (0.45) L3MBTL1LMNACRHR1MAPTALDH1A1
SCHEMBL7730352 0.82 MAPT (0.67) L3MBTL1LMNAMAPTPOLBALDH1A1
SCHEMBL7730097 0.82 LMNA (0.48) L3MBTL1LMNAMAPTPOLBALDH1A1
SCHEMBL7726527 0.81 CRHR1 (0.45) L3MBTL1LMNACRHR1ALDH1A1RAB9A
SCHEMBL7723511 0.80 MAPT (0.51) L3MBTL1LMNACRHR1MAPTPOLB
SCHEMBL7730095 0.79 MAPT (0.55) L3MBTL1LMNAMAPTPOLBKDM4E
SCHEMBL7724970 0.79 CRHR1 (0.49) L3MBTL1LMNACRHR1MAPTPOLB
SCHEMBL7723691 0.79 CRHR1 (0.49) L3MBTL1LMNACRHR1MAPTPOLB
SCHEMBL7723523 0.78 CRHR1 (0.51) L3MBTL1LMNACRHR1ALDH1A1KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6403586-B1 Pyridazine derivatives and drugs containing the same as the active ingredient KOWA CO., LTD. (JP) 2002-06-11 US disclosed
EP-1061077-A1 NOVEL PYRIDAZINE DERIVATIVES AND DRUGS CONTAINING THE SAME AS THE ACTIVE INGREDIENT Kowa Co., Ltd. (JP) 2000-12-20 EP disclosed