SCHEMBL7730488

SCHEMBL7730488

COc1c(NC(=O)c2coc([C@H](N)CCc3ccccc3)n2)cnc2ccccc12

nearest known ligand 0.40

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
BCHE P06276 11/20 0.40
MAPK1 P28482 1/20 0.37
NPC1 O15118 1/20 0.35
RAB9A P51151 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7732119 0.82 SLC2A1 (0.44)
SCHEMBL7732103 0.78 RAB9A (0.53) NPC1RAB9A
Trifluoroacetic Acid SCHEMBL7735917 0.74 RAB9A (0.48) NPC1RAB9A
SCHEMBL7732373 0.73 TRPV1 (0.50) NPC1RAB9A
SCHEMBL7732335 0.72 CES1 (0.49)
SCHEMBL7732052 0.72 RAB9A (0.43) NPC1RAB9A
SCHEMBL7733996 0.70 NPC1 (0.50) NPC1RAB9A
SCHEMBL7735550 0.69 TRPV1 (0.52) NPC1RAB9A
SCHEMBL7732173 0.68 TRPM8 (0.36) NPC1RAB9A
SCHEMBL7734013 0.67 NPC1 (0.45) NPC1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6436980-B1 TRANSPORT PROTEIN SUPPRESSORS; MICROBIOCIDES ESSENTIAL THERAPEUTICS, INC. 2002-08-20 US disclosed
US-6204279-B1 SECONDARY AMIDE CONTAINING BENZOXAZOLE DERIVATIVES MICROCIDE PHARMACEUTICALS, INC. 2001-03-20 US disclosed
WO-1999037667-A1 EFFLUX PUMP INHIBITORS MICROCIDE PHARMACEUTICALS, INC. (US) 1999-07-29 WO disclosed