SCHEMBL7733577

SCHEMBL7733577

Cc1cc2nc(C(O)[C@H](N)CC(C)C)oc2cc1C

nearest known ligand 0.45

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
AAK1 Q2M2I8 7/20 0.45
KDM4E B2RXH2 4/20 0.36
NPC1 O15118 4/20 0.36
ALDH1A1 P00352 4/20 0.36
RAB9A P51151 4/20 0.36
SMN1; SMN2 Q16637 4/20 0.36
HSD17B10 Q99714 4/20 0.36
KMT2A Q03164 1/20 0.36
TP53 P04637 4/20 0.33
MAPT P10636 3/20 0.33
HPGD P15428 3/20 0.33
GAA P10253 2/20 0.33
NPSR1 Q6W5P4 1/20 0.33
CHRNB2 P17787 1/20 0.32
CHRNA4 P43681 1/20 0.32
TAS1R3 Q7RTX0 4/20 0.31
TAS1R1 Q7RTX1 4/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7729637 0.77 METAP2 (0.41) KDM4ENPC1RAB9ASMN1; SMN2HSD17B10
SCHEMBL7722996 0.76 AAK1 (0.47) AAK1TP53MAPTCHRNB2CHRNA4
SCHEMBL7733987 0.76 AAK1 (0.38) AAK1TP53
SCHEMBL7732441 0.75 AAK1 (0.32) AAK1KDM4ENPC1ALDH1A1RAB9A
SCHEMBL7733548 0.74 AAK1 (0.46) AAK1NPC1RAB9AHSD17B10
SCHEMBL7730501 0.69 ALDH1A1 (0.46) AAK1KDM4EALDH1A1HSD17B10KMT2A
SCHEMBL8362696 0.69 ALDH1A1 (0.46) AAK1KDM4EALDH1A1HSD17B10KMT2A
SCHEMBL7733926 0.68 AAK1 (0.41) AAK1NPC1RAB9AKMT2AMAPT
SCHEMBL9305783 0.65 RAB9A (0.34) AAK1KDM4ENPC1ALDH1A1RAB9A
SCHEMBL9305778 0.64 RAB9A (0.38) KDM4ENPC1ALDH1A1RAB9ASMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6436980-B1 TRANSPORT PROTEIN SUPPRESSORS; MICROBIOCIDES ESSENTIAL THERAPEUTICS, INC. 2002-08-20 US disclosed
US-6204279-B1 SECONDARY AMIDE CONTAINING BENZOXAZOLE DERIVATIVES MICROCIDE PHARMACEUTICALS, INC. 2001-03-20 US disclosed