Fialuridine

Fialuridine

SCHEMBL773510

O=c1[nH]c(=O)n([C@@H]2O[C@H](CO)C(O)C2F)cc1I

nearest known ligand 0.77

Full drug profile on Sugi Atlas →

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
PYGM P11217 3/20 0.77
TK1 P04183 2/20 0.58
TK2 O00142 2/20 0.55
P2RY6 Q15077 5/20 0.52
P2RY14 Q15391 3/20 0.52
CDA P32320 1/20 0.47
SLC28A1 O00337 1/20 0.47
SLC28A2 O43868 1/20 0.47
SLC29A1 Q99808 1/20 0.47
SLC28A3 Q9HAS3 1/20 0.47
LMNA P02545 1/20 0.44
SMN1; SMN2 Q16637 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Fialuridine SCHEMBL1533997 1.00 PYGM (0.77) PYGMTK1TK2P2RY6P2RY14
Fialuridine SCHEMBL3084377 1.00 PYGM (0.77) PYGMTK1TK2P2RY6P2RY14
Fialuridine SCHEMBL30674 1.00 PYGM (0.77) PYGMTK1TK2P2RY6P2RY14
Fialuridine SCHEMBL13702050 1.00 PYGM (0.77) PYGMTK1TK2P2RY6P2RY14
Fialuridine SCHEMBL3084382 1.00 PYGM (0.77) PYGMTK1TK2P2RY6P2RY14
Fialuridine SCHEMBL9059414 1.00 PYGM (0.77) PYGMTK1TK2P2RY6P2RY14
Fialuridine SCHEMBL24359134 1.00 PYGM (0.77) PYGMTK1TK2P2RY6P2RY14
Fialuridine SCHEMBL768344 1.00 PYGM (0.77) PYGMTK1TK2P2RY6P2RY14
Fialuridine SCHEMBL20769829 1.00 PYGM (0.77) PYGMTK1TK2P2RY6P2RY14
Fialuridine SCHEMBL12658448 1.00 PYGM (0.77) PYGMTK1TK2P2RY6P2RY14

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 22 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-12397013-B2 Extrahepatic delivery ALNYLAM PHARMACEUTICALS, INC. (US) 2025-08-26 US disclosed
US-20240358738-A1 EXTRAHEPATIC DELIVERY BANK OF AMERICA, N.A. 2024-10-31 US disclosed
US-12005074-B2 Extrahepatic delivery ALNYLAM PHARMACEUTICALS, INC. (US) 2024-06-11 US disclosed
US-20240009225-A1 EXTRAHEPATIC DELIVERY BANK OF AMERICA, N.A. 2024-01-11 US disclosed
WO-2023220440-A1 OLIGONUCLEOTIDE COMPOSITIONS AND METHODS THEREOF WAVE LIFE SCIENCES LTD. (SG) 2023-11-16 WO disclosed
US-20220307024-A1 DELIVERY OF OLIGONUCLEOTIDES TO THE STRIATUM ALNYLAM PHARMACEUTICALS, INC. (US) 2022-09-29 US disclosed
US-20220125823-A1 EXTRAHEPATIC DELIVERY BANK OF AMERICA, N.A. 2022-04-28 US disclosed
EP-3983077-A1 DELIVERY OF OLIGONUCLEOTIDES TO THE STRIATUM Alnylam Pharmaceuticals, Inc. (US) 2022-04-20 EP disclosed
EP-3790970-A1 EXTRAHEPATIC DELIVERY Alnylam Pharmaceuticals Inc. (US) 2021-03-17 EP disclosed
WO-2020257194-A1 DELIVERY OF OLIGONUCLEOTIDES TO THE STRIATUM ALNYLAM PHARMACEUTICALS, INC. (US) 2020-12-24 WO disclosed
US-20190290670-A1 METHODS AND COMPOSITIONS FOR TREATING HEPATITIS C VIRUS IDENIX PHARMACEUTICALS LLC (US) 2019-09-26 US disclosed
US-10363265-B2 Methods and compositions for treating hepatitis C virus IDENIX PHARMACEUTICALS LLC (US) 2019-07-30 US disclosed
US-9968628-B2 Methods and compositions for treating flaviviruses and pestiviruses IDENIX PHARMACEUTICALS LLC (US) 2018-05-15 US disclosed
US-20130330297-A1 MODIFIED 2' AND 3'-NUCLEOSIDE PRODRUGS FOR TREATING FLAVIVIRIDAE INFECTIONS IDENIX PHARMACEUTICALS, INC. (US) 2013-12-12 US disclosed
US-8299038-B2 Methods and compositions for treating hepatitis C virus IDENIX PHARMACEUTICALS, INC. (US) 2012-10-30 US disclosed
US-20120071641-A1 NUCLEIC ACID CHEMICAL MODIFICATIONS ALNYLAM PHARMACEUTICALS, INC. (US) 2012-03-22 US disclosed
WO-2010101951-A1 NUCLEIC ACID CHEMICAL MODIFICATIONS ALNYLAM PHARMACEUTICALS, INC. (US) 2010-09-10 WO disclosed
US-20090280086-A1 METHODS AND COMPOSITIONS FOR TREATING HEPATITIS C VIRUS IDENIX PHARMACEUTICALS LLC 2009-11-12 US disclosed
US-7608600-B2 Treating hepatitis C virus infections; antivirals have low toxicity to the host; inhibit Flaviviridae polymerase IDENIX PHARMACEUTICALS, INC. (US) 2009-10-27 US disclosed
US-7608597-B2 Methods and compositions for treating hepatitis C virus IDENIX PHARMACEUTICALS, INC. (US) 2009-10-27 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (11 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20220307024-A1 DELIVERY OF OLIGONUCLEOTIDES TO THE STRIATUM SNRPE, AGO2, IGF2BP2 PYGM 2357/4885TK1 165/4885TK2 437/4885
US-20090280086-A1 METHODS AND COMPOSITIONS FOR TREATING HEPATITIS C VIRUS HAVCR2, HCCS, PYGL PYGM 198/4885TK1 143/4885TK2 396/4885
US-20240358738-A1 EXTRAHEPATIC DELIVERY RNASE1, SLC10A1, FABP1 PYGM 3618/4885TK1 134/4885TK2 258/4885
US-20190290670-A1 METHODS AND COMPOSITIONS FOR TREATING HEPATITIS C VIRUS HAVCR2, HCCS, PYGL PYGM 198/4885TK1 143/4885TK2 396/4885
US-12005074-B2 Extrahepatic delivery RNASE1, SLC10A1, FABP1 PYGM 3618/4885TK1 134/4885TK2 258/4885
US-10363265-B2 Methods and compositions for treating hepatitis C virus HAVCR2, HCCS, PYGL PYGM 198/4885TK1 143/4885TK2 396/4885
US-20220125823-A1 EXTRAHEPATIC DELIVERY RNASE1, LDLR, HAVCR2 PYGM 3715/4885TK1 172/4885TK2 309/4885
US-20240009225-A1 EXTRAHEPATIC DELIVERY RNASE1, SLC10A1, FABP1 PYGM 3618/4885TK1 134/4885TK2 258/4885
US-20130330297-A1 MODIFIED 2' AND 3'-NUCLEOSIDE PRODRUGS FOR TREATING FLAVIVIRIDAE INFECTIONS PNP, UGT1A3, UGT2B7 PYGM 411/4885TK1 124/4885TK2 177/4885
US-12397013-B2 Extrahepatic delivery RNASE1, LDLR, HAVCR2 PYGM 3715/4885TK1 172/4885TK2 309/4885
US-20120071641-A1 NUCLEIC ACID CHEMICAL MODIFICATIONS NSUN2, RNMT, NSUN3 PYGM 3144/4885TK1 155/4885TK2 219/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.