SCHEMBL7737834

SCHEMBL7737834

O=C(O)COc1cccc2c1OCC(=O)N2CCO

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTGIR P43119 1/20 0.43
ALDH1A1 P00352 4/20 0.39
HTR6 P50406 1/20 0.38
PTGDR2 Q9Y5Y4 3/20 0.38
KDM4E B2RXH2 2/20 0.38
HPGD P15428 2/20 0.38
TDP1 Q9NUW8 1/20 0.38
KMO O15229 2/20 0.38
DRD2 P14416 2/20 0.38
HTR2A P28223 2/20 0.38
MCHR1 Q99705 2/20 0.38
POLB P06746 1/20 0.37
SMN1; SMN2 Q16637 1/20 0.37
GLA P06280 1/20 0.37
L3MBTL1 Q9Y468 1/20 0.37
MEN1 O00255 1/20 0.35
KMT2A Q03164 1/20 0.35
ALOX12 P18054 1/20 0.35
CHRM2 P08172 1/20 0.35
CHRM4 P08173 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7736555 0.82 PTGIR (0.47) PTGIRALDH1A1HTR6DRD2HTR2A
SCHEMBL7737346 0.81 PTGIR (0.49) PTGIRALDH1A1DRD2HTR2AMCHR1
SCHEMBL7739689 0.81 ALOX12 (0.40) ALDH1A1HTR6HPGDKMODRD2
SCHEMBL7730040 0.79 ALOX12 (0.53) ALDH1A1KDM4EHPGDL3MBTL1MEN1
SCHEMBL7736507 0.77 PTGIR (0.63) PTGIRALDH1A1PTGDR2KDM4EHPGD
SCHEMBL7729988 0.77 HTR6 (0.41) ALDH1A1HTR6KMODRD2HTR2A
SCHEMBL3584551 0.76 HTR6 (0.41) ALDH1A1HTR6KMODRD2HTR2A
SCHEMBL7737250 0.72 PTGIR (0.46) PTGIRPTGDR2ALOX12
SCHEMBL7522216 0.71 PARP1 (0.50) ALDH1A1PTGDR2KDM4EHPGDTDP1
SCHEMBL7736480 0.71 ALDH1A1 (0.41) ALDH1A1POLBMEN1KMT2ACHRM1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6407096-B1 1,4-BENZOTHIAZINE AND 1,4-BENZOXAZINE DERIVATIVES; HYPOTENSIVE, ANTIISCHEMIC, ANTIALLERGEN, ANTIASTHMATIC AND ANTICOAGULANT AGENTS; CARDIOVASCULAR DISORDERS TORAY INDUSTRIES, INC. (JP) 2002-06-18 US disclosed
EP-1028113-A1 FUSED BENZENE HETEROCYCLE DERIVATIVES AND UTILIZATION THEREOF TORAY INDUSTRIES, INC. (JP) 2000-08-16 EP disclosed