SCHEMBL7729988

SCHEMBL7729988

O=C1COc2c(O)cccc2N1CCO

nearest known ligand 0.41

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
HTR6 P50406 1/20 0.41
ALDH1A1 P00352 2/20 0.40
DRD4 P21917 1/20 0.38
DRD2 P14416 3/20 0.38
HTR2A P28223 3/20 0.38
MCHR1 Q99705 2/20 0.38
CHRM1 P11229 2/20 0.37
MEN1 O00255 2/20 0.36
KMT2A Q03164 2/20 0.36
KMO O15229 1/20 0.36
USP2 O75604 1/20 0.36
CYP2D6 P10635 1/20 0.36
TSHR P16473 2/20 0.36
GAA P10253 1/20 0.36
TP53 P04637 1/20 0.36
HEXA P06865 1/20 0.36
HEXB P07686 1/20 0.36
HTR1A P08908 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3584551 0.84 HTR6 (0.41) HTR6ALDH1A1DRD4DRD2HTR2A
SCHEMBL7737728 0.79 HTR6 (0.45) HTR6ALDH1A1DRD4DRD2HTR2A
SCHEMBL7358743 0.77 ALDH1A1 (0.61) ALDH1A1DRD4MEN1KMT2AUSP2
SCHEMBL7737834 0.77 PTGIR (0.43) HTR6ALDH1A1DRD2HTR2AMCHR1
SCHEMBL7737187 0.77 HTR6 (0.41) HTR6ALDH1A1DRD2HTR2AMCHR1
SCHEMBL7739689 0.74 ALOX12 (0.40) HTR6ALDH1A1DRD2HTR2AMCHR1
SCHEMBL7736480 0.74 ALDH1A1 (0.41) ALDH1A1CHRM1MEN1KMT2ATSHR
SCHEMBL13545339 0.73 CHRM1 (0.42) HTR6DRD2HTR2AMCHR1CHRM1
SCHEMBL7730055 0.72 ALOX12 (0.58) ALDH1A1MEN1KMT2AGAATP53
SCHEMBL7729866 0.70 DRD2 (0.38) DRD4DRD2HTR2AKMT2ATSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1202084-C Fused benzene heterocycle derivatives and utilization thereof TORAY INDUSTRIES (JP) 2005-05-18 CN disclosed
US-6407096-B1 1,4-BENZOTHIAZINE AND 1,4-BENZOXAZINE DERIVATIVES; HYPOTENSIVE, ANTIISCHEMIC, ANTIALLERGEN, ANTIASTHMATIC AND ANTICOAGULANT AGENTS; CARDIOVASCULAR DISORDERS TORAY INDUSTRIES, INC. (JP) 2002-06-18 US disclosed
CN-1287553-A Fused benzene heterocycle derivatives and utilization thereof TORAY INDUSTRIES (JP) 2001-03-14 CN disclosed
EP-1028113-A1 FUSED BENZENE HETEROCYCLE DERIVATIVES AND UTILIZATION THEREOF TORAY INDUSTRIES, INC. (JP) 2000-08-16 EP disclosed