SCHEMBL7740420

SCHEMBL7740420

CC(C)(C)OC(=O)C(N)c1cc(NC(N)=S)ccc1-n1cccn1

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SYK P43405 1/20 0.37
ALDH1A1 P00352 8/20 0.37
MEN1 O00255 7/20 0.37
KMT2A Q03164 7/20 0.37
MAPT P10636 6/20 0.37
LMNA P02545 3/20 0.37
RAB9A P51151 1/20 0.37
NPSR1 Q6W5P4 1/20 0.37
RXFP1 Q9HBX9 1/20 0.36
KCNH2 Q12809 2/20 0.35
HTT P42858 1/20 0.34
MDM2 Q00987 1/20 0.34
L3MBTL1 Q9Y468 1/20 0.34
CYP2C8 P10632 1/20 0.33
CYP2C9 P11712 1/20 0.33
GAA P10253 1/20 0.33
LRRK2 Q5S007 1/20 0.32
KDM4E B2RXH2 1/20 0.32
HPGD P15428 1/20 0.32
IDH2 P48735 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27525664 0.83 RXFP1 (0.35) SYKALDH1A1MEN1KMT2AMAPT
SCHEMBL27493987 0.80 ALDH1A1 (0.33) SYKALDH1A1MEN1KMT2AMAPT
SCHEMBL7740422 0.78 SYK (0.40) SYKALDH1A1MEN1KMT2AMAPT
SCHEMBL22044797 0.76 NR1I3 (0.43) SYKALDH1A1MEN1KMT2AMAPT
SCHEMBL27506223 0.72 ALDH1A1 (0.49) ALDH1A1MEN1KMT2AMAPTLMNA
SCHEMBL22044738 0.70 NAMPT (0.44) SYKALDH1A1MEN1KMT2AMAPT
SCHEMBL27564255 0.68 NTRK1 (0.31)
SCHEMBL27495566 0.68 GPR119 (0.35) KCNH2CYP2C8CYP2C9
SCHEMBL7738864 0.67 SYK (0.35) SYKALDH1A1MEN1KMT2AMAPT
SCHEMBL7734196 0.67 HDAC3 (0.32) ALDH1A1MEN1KMT2AMAPTLMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1217928-C Heterocyclic compound having NOS inhibitory action CHUGAI SEIYAKA K K (JP) 2005-09-07 CN disclosed
US-6414005-B1 BRAIN DISORDERS; ALZHEIMER'S DISEASE; PARKINSON'S DISEASE CHUGAI SEIYAKU KABUSHIKI KAISHA (JP) 2002-07-02 US disclosed
CN-1280565-A Heterocyclic compounds having NOS inhibitory activities CHUGAI SEIYAKA K K (JP) 2001-01-17 CN disclosed
EP-1043312-A1 HETEROCYCLIC COMPOUNDS HAVING NOS INHIBITORY ACTIVITIES CHUGAI SEIYAKU KABUSHIKI KAISHA (JP) 2000-10-11 EP disclosed