SCHEMBL27564255

SCHEMBL27564255

CCSC(=N)Nc1ccc(-n2cc(C)cn2)c(C(N)C(=O)OC(C)(C)C)c1

nearest known ligand 0.31

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
NTRK1 P04629 1/20 0.31
PIK3CA P42336 1/20 0.31
PIK3CG P48736 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27525664 0.85 RXFP1 (0.35)
Hydrochloric Acid SCHEMBL27512818 0.75 TDO2 (0.32) NTRK1PIK3CAPIK3CG
Hydrochloric Acid SCHEMBL7740435 0.75 TDO2 (0.32) NTRK1PIK3CAPIK3CG
SCHEMBL7734196 0.70 HDAC3 (0.32)
SCHEMBL7740420 0.68 SYK (0.37)
SCHEMBL7734182 0.65 GRM2 (0.33) NTRK1PIK3CAPIK3CG
SCHEMBL7740424 0.65 MEN1 (0.36)
SCHEMBL8116723 0.65 TDO2 (0.33) NTRK1PIK3CAPIK3CG
SCHEMBL7734178 0.64 NTRK1 (0.35) NTRK1PIK3CAPIK3CG
SCHEMBL7740476 0.64 NOS1 (0.38)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1217928-C Heterocyclic compound having NOS inhibitory action CHUGAI SEIYAKA K K (JP) 2005-09-07 CN disclosed
CN-1280565-A Heterocyclic compounds having NOS inhibitory activities CHUGAI SEIYAKA K K (JP) 2001-01-17 CN disclosed