SCHEMBL7741874

SCHEMBL7741874

CC[C@@H]1C(=O)O[C@H]2[C@H]1CC/C(C)=C/CC[C@@]1(C)O[C@@H]21

nearest known ligand 0.73

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.56
NLRP3 Q96P20 4/20 0.56
PKM P14618 4/20 0.56
LMNA P02545 3/20 0.56
TP53 P04637 3/20 0.56
CYP3A4 P08684 3/20 0.56
NFKB1 P19838 2/20 0.56
CYP1A2 P05177 2/20 0.56
STAT6 P42226 2/20 0.56
MAPT P10636 2/20 0.56
CASP1 P29466 1/20 0.56
PTGS2 P35354 1/20 0.56
NFKB2 Q00653 1/20 0.56
RELA Q04206 1/20 0.56
CYP2D6 P10635 1/20 0.56
TSHR P16473 1/20 0.56
MAPK1 P28482 1/20 0.56
THPO P40225 1/20 0.56
HTT P42858 1/20 0.56
HIF1A Q16665 1/20 0.56

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13251201 1.00 ALDH1A1 (0.56) ALDH1A1NLRP3PKMLMNATP53
SCHEMBL13433133 0.91 PKM (0.54) ALDH1A1NLRP3PKMLMNATP53
SCHEMBL16421406 0.90 ALDH1A1 (0.55) ALDH1A1NLRP3PKMLMNATP53
SCHEMBL17761701 0.90 ALDH1A1 (0.55) ALDH1A1NLRP3PKMLMNATP53
SCHEMBL15336431 0.90 ALDH1A1 (0.55) ALDH1A1NLRP3PKMLMNATP53
Dimethylaminoparthenolide SCHEMBL6741648 0.89 NLRP3 (0.54) ALDH1A1NLRP3PKMLMNATP53
Dimethylaminoparthenolide SCHEMBL16414703 0.89 NLRP3 (0.54) ALDH1A1NLRP3PKMLMNATP53
Dimethylaminoparthenolide SCHEMBL29496871 0.89 NLRP3 (0.54) ALDH1A1NLRP3PKMLMNATP53
Dimethylaminoparthenolide SCHEMBL10099623 0.89 NLRP3 (0.54) ALDH1A1NLRP3PKMLMNATP53
Dimethylaminoparthenolide SCHEMBL16414642 0.89 NLRP3 (0.54) ALDH1A1NLRP3PKMLMNATP53

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9512138-B2 Compositions and methods for treating cancer THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 2016-12-06 US disclosed
US-9512138-B2 Compositions and methods for treating cancer THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 2016-12-06 US disclosed
US-20160137662-A1 COMPOSITIONS AND METHODS FOR TREATING CANCER THE GOVERNMENT OF THE UNITED STATES, AS REPRESENTED BY THE SECRETARY OF THE ARMY 2016-05-19 US disclosed
US-20160137662-A1 COMPOSITIONS AND METHODS FOR TREATING CANCER THE GOVERNMENT OF THE UNITED STATES, AS REPRESENTED BY THE SECRETARY OF THE ARMY 2016-05-19 US disclosed
US-20150031725-A1 COMPOSITIONS AND METHODS FOR TREATING CANCER THE REGENTS OF THE UNIVERSITY OF CALIFORNIA 2015-01-29 US disclosed
US-20100009970-A1 COMPOSITIONS AND METHODS FOR TREATMENT OF VIRAL DISEASES COMBINATORX (SINGAPORE) PTE. LTD. (SG) 2010-01-14 US disclosed
US-20080161324-A1 Compositions and methods for treatment of viral diseases EXCRX (SINGAPORE) PTE. LTD. (F.K.A. COMBINATORX (SINGAPORE) PTE LTD.) (SG) 2008-07-03 US disclosed
US-7312242-B2 Use of parthenolide derivatives as antileukemic and cytotoxic agents UNIVERSITY OF KENTUCKY (US) 2007-12-25 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (4 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20160137662-A1 COMPOSITIONS AND METHODS FOR TREATING CANCER HRAS, TP53, VHL ALDH1A1 2822/4885NLRP3 4049/4885PKM 2957/4885
US-20100009970-A1 COMPOSITIONS AND METHODS FOR TREATMENT OF VIRAL DISEASES HTR1A, HTR3B, HTR3A ALDH1A1 2240/4885NLRP3 1644/4885PKM 1577/4885
US-20150031725-A1 COMPOSITIONS AND METHODS FOR TREATING CANCER HRAS, TP53, VHL ALDH1A1 2822/4885NLRP3 4049/4885PKM 2957/4885
US-20080161324-A1 Compositions and methods for treatment of viral diseases HAVCR2, EIF2AK2, RNASE1 ALDH1A1 785/4885NLRP3 1562/4885PKM 2372/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.