SCHEMBL7742013

SCHEMBL7742013

CCCCOC(=O)[C@@H](CC(N)=O)NC(=O)OCc1ccccc1

nearest known ligand 0.55

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
CTSL P07711 3/20 0.55
CTSS P25774 3/20 0.55
PSMB1 P20618 1/20 0.53
SIRT2 Q8IXJ6 3/20 0.52
ALDH1A1 P00352 1/20 0.51
CYP3A4 P08684 1/20 0.51
TSHR P16473 1/20 0.51
MAPK1 P28482 1/20 0.51
TDP1 Q9NUW8 1/20 0.51
L3MBTL1 Q9Y468 1/20 0.51
CTSK P43235 6/20 0.50
ITGB3 P05106 4/20 0.49
ITGA2B P08514 4/20 0.49
CASP1 P29466 1/20 0.49
PSMB8 P28062 1/20 0.48
PSMB5 P28074 1/20 0.48
SIRT1 Q96EB6 2/20 0.48
SIRT3 Q9NTG7 1/20 0.48
CTSB P07858 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7742011 1.00 CTSL (0.55) CTSLCTSSPSMB1SIRT2ALDH1A1
SCHEMBL22975021 0.88 CTSL (0.57) CTSLCTSSSIRT2ALDH1A1CYP3A4
SCHEMBL28678129 0.88 CTSL (0.57) CTSLCTSSSIRT2ALDH1A1CYP3A4
SCHEMBL7742003 0.88 PSMB1 (0.56) CTSLCTSSPSMB1ALDH1A1CTSK
SCHEMBL7742845 0.88 PSMB1 (0.56) CTSLCTSSPSMB1ALDH1A1CTSK
SCHEMBL7688519 0.87 PSMB1 (0.57) CTSLCTSSPSMB1CTSKCASP1
Hydrochloric Acid SCHEMBL29604804 0.87 CTSL (0.56) CTSLCTSSSIRT2ALDH1A1CYP3A4
SCHEMBL2026643 0.86 SIRT2 (0.52) CTSLCTSSPSMB1SIRT2ALDH1A1
SCHEMBL6254290 0.85 CASP1 (0.57) CTSLCTSSALDH1A1CYP3A4TSHR
SCHEMBL4452037 0.85 CASP1 (0.57) CTSLCTSSALDH1A1CYP3A4TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6420166-B2 REACTING AN N-PROTECTED ASPARAGINE ESTER WITH A PROTEASE IN AQUEOUS SOLUTION AT PH OF 6.0 TO 7.5 AND AN ORGANIC SOLVENT, AND EXTRACTING THE N-PROTECTED-D-ASPARAGINE ESTER; CHEMICAL INTERMEDIATES TO ANTIBACTERIAL COMPOUNDS BASOLEA PHARMACEUTICA AG (CH) 2002-07-16 US disclosed
US-20010049127-A1 Process for the preparation of D-asparagine derivatives HOFFMANN-LA ROCHE INC. 2001-12-06 US disclosed
EP-1148140-A1 Process for the preparation of D-asparagine derivatives Basilea Pharmaceutica AG (CH) 2001-10-24 EP disclosed