SCHEMBL7743869

SCHEMBL7743869

O=C(OC[C@H]1O[C@@H](n2cnc3c(NCc4cccc(I)c4)nc(Cl)nc32)[C@H](OC(=O)c2ccccc2)[C@@H]1OC(=O)c1ccccc1)c1ccccc1

nearest known ligand 0.66

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
ADORA3 P0DMS8 17/20 0.66
ADORA1 P30542 6/20 0.66
ADORA2A P29274 5/20 0.66
ADORA2B P29275 1/20 0.61
HTR2C P28335 1/20 0.58
PPARG P37231 1/20 0.58
HTR2B P41595 1/20 0.58
PPARD Q03181 1/20 0.58
ABCG2 Q9UNQ0 1/20 0.58
TP53 P04637 1/20 0.58
CYP1A2 P05177 1/20 0.58
MAPT P10636 1/20 0.58
MAPK1 P28482 1/20 0.58

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24601182 0.88 ADORA3 (0.78) ADORA3ADORA1ADORA2AADORA2BHTR2C
SCHEMBL19370184 0.86 NT5E (0.65) ADORA3ADORA1ADORA2A
SCHEMBL8327419 0.85 ALDH1A1 (0.53) ADORA3ADORA1ADORA2AADORA2BTP53
SCHEMBL7744287 0.84 ADORA3 (0.62) ADORA3ADORA1ADORA2AADORA2BHTR2C
SCHEMBL9404051 0.84 ALDH1A1 (0.51) ADORA3ADORA1ADORA2ATP53MAPT
SCHEMBL8819182 0.84 ALDH1A1 (0.51) ADORA3ADORA1ADORA2ATP53MAPT
SCHEMBL8820179 0.83 ALDH1A1 (0.50) ADORA3ADORA1ADORA2ATP53MAPT
SCHEMBL23436497 0.82 LMNA (0.69) TP53MAPT
SCHEMBL8818839 0.82 LMNA (0.69) TP53MAPT
SCHEMBL15679138 0.82 LMNA (0.69) TP53MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0708781-B1 A 3 ADENOSINE RECEPTOR AGONISTS USA (US) 2001-10-04 EP disclosed
EP-0708781-A1 A 3 ADENOSINE RECEPTOR AGONISTS THE UNITED STATES OF AMERICA, as represented by THE SECRETARY, Department of Health and Human Services (US) 1996-05-01 EP disclosed
WO-1995002604-A1 A3 ADENOSINE RECEPTOR AGONISTS THE UNITED STATES OF AMERICA, REPRESENTED BY THE SECRETARY, DEPARTMENT OF HEALTH AND HUMAN SERVICES (US) 1995-01-26 WO disclosed