SCHEMBL7744137

SCHEMBL7744137

CC[C@H](C)N1C(=O)C(C(C(N)=O)c2ccc(C(F)(F)F)cc2C(F)(F)F)C=C(c2ccccc2)c2ccccc21

nearest known ligand 0.36

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 1/20 0.36
NOTCH1 P46531 4/20 0.35
NOTCH3 Q9UM47 4/20 0.35
PPARG P37231 2/20 0.34
GALR3 O60755 1/20 0.34
CYP2C9 P11712 1/20 0.33
SCN9A Q15858 1/20 0.33
CCKBR P32239 4/20 0.33
CCKAR P32238 2/20 0.33
F7 P08709 1/20 0.33
EDNRB P24530 1/20 0.33
EDNRA P25101 1/20 0.33
AKR1C3 P42330 1/20 0.33
AKR1C2 P52895 1/20 0.33
PDE2A O00408 1/20 0.32
P2RX4 Q99571 1/20 0.32
FPR2 P25090 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7738908 0.84 KCNH2 (0.45) KCNH2NOTCH1NOTCH3CCKBRCCKAR
SCHEMBL7744132 0.70 KCNH2 (0.45) KCNH2NOTCH1NOTCH3CCKBRCCKAR
SCHEMBL7744591 0.70 KCNH2 (0.45) KCNH2NOTCH1NOTCH3CCKBRCCKAR
SCHEMBL7744135 0.69 KCNH2 (0.72) KCNH2NOTCH1NOTCH3CCKBRCCKAR
SCHEMBL7744698 0.67 KCNH2 (0.47) KCNH2GALR3SCN9AFPR2
SCHEMBL7744588 0.66 CCKBR (0.44) KCNH2NOTCH1NOTCH3CCKBR
SCHEMBL7744124 0.65 KCNH2 (0.55) KCNH2CCKBRCCKAR
SCHEMBL7743995 0.65 KCNH2 (0.36) KCNH2GALR3SCN9ACCKBRCCKAR
SCHEMBL18243407 0.60 PDE2A (0.49) CYP2C9F7PDE2A
SCHEMBL30428378 0.59 CES2 (0.50) F7AKR1C3AKR1C2PDE2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2001010216-A1 ANTIARRHYTHMIC COMPOUNDS MERCK & CO., INC. (US) 2001-02-15 WO disclosed