SCHEMBL7744286

SCHEMBL7744286

CC(=O)NN1CN([C@@H]2O[C@H](CO)C(O)C2O)c2ncnc(O)c21

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.39
MAPK1 P28482 2/20 0.39
TDP1 Q9NUW8 2/20 0.39
KDM4E B2RXH2 2/20 0.39
HTT P42858 2/20 0.39
HIF1A Q16665 2/20 0.39
CYP1A2 P05177 1/20 0.39
STAT6 P42226 1/20 0.39
TP53 P04637 1/20 0.39
ALOX15 P16050 1/20 0.39
HSD17B10 Q99714 1/20 0.39
HDAC6 Q9UBN7 1/20 0.39
SMN1; SMN2 Q16637 3/20 0.39
TSHR P16473 2/20 0.39
GAA P10253 1/20 0.39
BLM P54132 1/20 0.39
CDA P32320 2/20 0.38
ADORA1 P30542 2/20 0.38
SLC29A1 Q99808 1/20 0.38
HSPA8 P11142 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7744270 0.90 MAPK1 (0.40) ALDH1A1MAPK1TDP1KDM4EHTT
SCHEMBL1976100 0.89 HSPA8 (0.46) ALDH1A1MAPK1TDP1KDM4EHTT
SCHEMBL453483 0.81 MAPK1 (0.46) ALDH1A1MAPK1TDP1KDM4EHTT
SCHEMBL453482 0.81 MAPK1 (0.46) ALDH1A1MAPK1TDP1KDM4EHTT
SCHEMBL177666 0.79 HSPA8 (0.44) ALDH1A1MAPK1TDP1KDM4EHTT
SCHEMBL6636043 0.77 MAPK1 (0.38) ALDH1A1MAPK1TDP1KDM4EHTT
SCHEMBL7617960 0.77 ADORA3 (0.43) ALDH1A1MAPK1TDP1KDM4EHTT
SCHEMBL8804156 0.75 KDM4E (0.38) ALDH1A1MAPK1TDP1KDM4EHTT
SCHEMBL9243746 0.75 ADORA1 (0.39) ALDH1A1MAPK1TDP1KDM4EHTT
SCHEMBL7746161 0.75 HSPA8 (0.42) MAPK1HIF1ASTAT6SMN1; SMN2ADORA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0708781-B1 A 3 ADENOSINE RECEPTOR AGONISTS USA (US) 2001-10-04 EP disclosed
US-5773423-A XANTHINE RIBOSIDES THE UNITED STATES OF AMERICA AS REPRESENTED BY THE DEPARTMENT OF HEALTH AND HUMAN SERVICES (US) 1998-06-30 US disclosed
EP-0708781-A1 A 3 ADENOSINE RECEPTOR AGONISTS THE UNITED STATES OF AMERICA, as represented by THE SECRETARY, Department of Health and Human Services (US) 1996-05-01 EP disclosed
WO-1995002604-A1 A3 ADENOSINE RECEPTOR AGONISTS THE UNITED STATES OF AMERICA, REPRESENTED BY THE SECRETARY, DEPARTMENT OF HEALTH AND HUMAN SERVICES (US) 1995-01-26 WO disclosed