SCHEMBL7752945

SCHEMBL7752945

CCc1ccc2c(c1)C(CCN)CO2

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR1A P08908 2/20 0.58
HTR2C P28335 2/20 0.58
HTR1D P28221 1/20 0.58
HCRTR2 O43614 1/20 0.41
PARP1 P09874 1/20 0.36
TAAR1 Q96RJ0 4/20 0.35
MAOB P27338 1/20 0.33
SLC6A2 P23975 3/20 0.33
SLC6A4 P31645 3/20 0.33
SLC6A3 Q01959 2/20 0.33
MEN1 O00255 3/20 0.32
KMT2A Q03164 3/20 0.32
MAPT P10636 2/20 0.32
CYP3A4 P08684 1/20 0.32
SMN1; SMN2 Q16637 1/20 0.32
RAB9A P51151 1/20 0.32
HTR2B P41595 1/20 0.31
SIGMAR1 Q99720 1/20 0.31
TP53 P04637 1/20 0.31
KIF11 P52732 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7752947 0.88 HTR1A (0.56) HTR1AHTR2CHTR1DHCRTR2TAAR1
SCHEMBL7757639 0.86 HTR2C (0.53) HTR1AHTR2CHTR1DTAAR1SLC6A2
SCHEMBL95790 0.81 HTR2C (0.61) HTR1AHTR2CHTR1DHCRTR2SLC6A2
SCHEMBL8130244 0.78 HTR1A (0.57) HTR1AHTR2CHTR1DTAAR1TP53
SCHEMBL172889 0.78 HTR1A (0.57) HTR1AHTR2CHTR1DHCRTR2MEN1
SCHEMBL7757152 0.77 MTNR1A (0.50) HTR1AHTR2CHTR1DHCRTR2MEN1
SCHEMBL13038051 0.76 HCRTR2 (0.48) HCRTR2PARP1CYP3A4TP53
SCHEMBL22923302 0.76 HCRTR2 (0.48) HCRTR2PARP1CYP3A4TP53
SCHEMBL6215060 0.75 HTR1A (0.57) HTR1AHTR2CHTR1DHCRTR2
SCHEMBL6339887 0.74 HTR1A (0.55) HTR1AHTR2CHTR1DMAOBSLC6A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0721947-B1 Alkyl(hetero)cyclic compounds, process for their preparation and pharmaceutical compositions containing them ADIR (FR) 2001-03-14 EP disclosed
US-5703121-A SLEEP DISORDERS ADIR ET COMPAGNIE (FR) 1997-12-30 US disclosed
EP-0721947-A1 Alkyl(hetero)cyclic compounds, process for their preparation and pharmaceutical compositions containing them ADIR ET COMPAGNIE (FR) 1996-07-17 EP disclosed