Nyasol

Nyasol

SCHEMBL776219

C=CC(/C=C/c1ccc(O)cc1)c1ccc(O)cc1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Full drug profile on Sugi Atlas →

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
APP P05067 5/20 0.43
ESR1 P03372 4/20 0.42
ESR2 Q92731 3/20 0.42
MAOB P27338 3/20 0.41
AKR1B1 P15121 3/20 0.41
PTGS2 P35354 2/20 0.41
AKR1B10 O60218 2/20 0.41
GLO1 Q04760 1/20 0.41
CAMK2A Q9UQM7 1/20 0.41
KDM4E B2RXH2 3/20 0.41
ALDH1A1 P00352 3/20 0.41
MAPT P10636 3/20 0.41
CYP2C9 P11712 3/20 0.41
CA12 O43570 3/20 0.41
CA1 P00915 3/20 0.41
CA2 P00918 3/20 0.41
CA3 P07451 3/20 0.41
CA4 P22748 3/20 0.41
CA6 P23280 3/20 0.41
CA5A P35218 3/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Nyasol SCHEMBL8416158 1.00 APP (0.43) APPESR1ESR2MAOBAKR1B1
Nyasol SCHEMBL776218 1.00 APP (0.43) APPESR1ESR2MAOBAKR1B1
Nyasol SCHEMBL799383 1.00 APP (0.43) APPESR1ESR2MAOBAKR1B1
Nyasol SCHEMBL30712027 1.00 APP (0.43) APPESR1ESR2MAOBAKR1B1
SCHEMBL13558420 0.92 CYP3A4 (0.46) APPESR1ESR2MAOBAKR1B1
SCHEMBL7861271 0.92 CYP3A4 (0.46) APPESR1ESR2MAOBAKR1B1
SCHEMBL799612 0.90 MAOB (0.39) APPESR1ESR2MAOBAKR1B1
SCHEMBL805124 0.87 MAPT (0.50) ESR2PTGS2KDM4EALDH1A1MAPT
SCHEMBL7861615 0.87 MAPT (0.50) ESR2PTGS2KDM4EALDH1A1MAPT
SCHEMBL7864584 0.87 MAPT (0.50) ESR2PTGS2KDM4EALDH1A1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 72 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20250195452-A1 ER-BETA ESTROGENIC COMPOUNDS AND METHODS OF USE IATERION, INC. 2025-06-19 US claimed
EP-4561582-A1 ER-BETA ESTROGENIC COMPOUNDS AND METHODS OF USE Iaterion, Inc. (US) 2025-06-04 EP claimed
WO-2024026037-A1 ER-BETA ESTROGENIC COMPOUNDS AND METHODS OF USE IATERION, INC. (US) 2024-02-01 WO claimed
US-20120277169-A1 NYASOL AND ANALOGS THEREOF FOR THE TREATMENT OF ESTROGEN RECEPTOR BETA-MEDIATED DISEASES BIONOVO, INC. (US) 2012-11-01 US claimed
US-20120070515-A1 Composition Comprising the Extract of Anemarrhena Asphodeloides Bunge or the Compounds Isolated from the Same for Preventing and Treating Lipid Metabolism Disorder EWHA UNIVERSITY- INDUSTRY COLLABORATION FOUNDATION (KR) 2012-03-22 US claimed
EP-2323641-A2 NYASOL AND ANALOGS THEREOF FOR THE TREATMENT OF ESTROGEN RECEPTOR BETA-MEDIATED DISEASES Bionovo Inc. (US) 2011-05-25 EP claimed
EP-2310024-A2 ESTROGENIC EXTRACTS FOR USE IN TREATING VAGINAL AND VULVAR ATROPHY Bionovo Inc. (US) 2011-04-20 EP claimed
WO-2010120029-A1 COMPOSITION COMPRISING THE EXTRACT OF ANEMARRHENA ASPHODELOIDES BUNGE OR THE COMPOUNDS ISOLATED FROM THE SAME FOR PREVENTING AND TREATING LIPID METABOLISM DISORDER EWHA UNIVERSITY - INDUSTRY COLLABORATION FOUNDATION (KR) 2010-10-21 WO claimed
WO-2010053600-A2 NYASOL AND ANALOGS THEREOF FOR THE TREATMENT OF ESTROGEN RECEPTOR BETA-MEDIATED DISEASES BIONOVO, INC. (US) 2010-05-14 WO claimed
US-20090312274-A1 Nyasol and Analogs Thereof for the Treatment of Estrogen Receptor Beta-Mediated Diseases BIONOVO, INC. (US) 2009-12-17 US claimed
US-20090304825-A1 ESTROGENIC EXTRACTS FOR USE IN TREATING VAGINAL AND VULVAR ATROPHY BIONOVO, INC. (US) 2009-12-10 US claimed
WO-2009137534-A2 ESTROGENIC EXTRACTS FOR USE IN TREATING VAGINAL AND VULVAR ATROPHY BIONOVO, INC. (US) 2009-11-12 WO claimed
JP-9301856-A None JP disclosed
US-20250213593-A1 Use of Derivatives based on Sarsasapogenin Structure and Pharmaceutical Compositions thereof BEIJING PHYTOVENT PHARMACEUTICAL TECHNOLOGY CO., LTD. (CN) 2025-07-03 US disclosed
US-20250195452-A1 ER-BETA ESTROGENIC COMPOUNDS AND METHODS OF USE IATERION, INC. 2025-06-19 US disclosed
EP-4561582-A1 ER-BETA ESTROGENIC COMPOUNDS AND METHODS OF USE Iaterion, Inc. (US) 2025-06-04 EP disclosed
EP-0925598-A1 COLOR DISPLAY DEVICE HAVING COLOR FILTER LAYERS Koninklijke Philips Electronics N.V. (NL) 1999-06-30 EP disclosed
WO-1998054742-A1 COLOR DISPLAY DEVICE HAVING COLOR FILTER LAYERS KONINKLIJKE PHILIPS ELECTRONICS N.V. (NL) 1998-12-03 WO disclosed
JP-H09301856-A ESTROGENIC AGENT JUMOKU SEIRI KINOUSEI BUTSUSHITSU GIJUTSU KENKYU KUMIAI 1997-11-25 JP disclosed
US-4876348-A DEHYDROCYCLIZATION OF 2-METHYLGLUTARONITRILE, AMMOXIDATION OF REACTION MIXTURE OVER MIXED OXIDE CATALYST THE STANDARD OIL COMPANY (US) 1989-10-24 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (6 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20090312274-A1 Nyasol and Analogs Thereof for the Treatment of Estrogen Receptor Beta-Mediated Diseases ESR2, ESR1, ESRRA APP 3260/4885ESR1 2/4885ESR2 1/4885
US-20120277169-A1 NYASOL AND ANALOGS THEREOF FOR THE TREATMENT OF ESTROGEN RECEPTOR BETA-MEDIATED DISEASES ESR2, ESR1, ESRRA APP 3260/4885ESR1 2/4885ESR2 1/4885
US-20250195452-A1 ER-BETA ESTROGENIC COMPOUNDS AND METHODS OF USE ESR2, ESR1, ESRRB APP 722/4885ESR1 2/4885ESR2 1/4885
US-20250213593-A1 Use of Derivatives based on Sarsasapogenin Structure and Pharmaceutical Compositions thereof MAVS, NLN, TFAM APP 326/4885ESR1 4720/4885ESR2 4151/4885
US-20120070515-A1 Composition Comprising the Extract of Anemarrhena Asphodeloides Bunge or the Compounds Isolated from the Same for Preventing and Treating Lipid Metabolism Disorder FABP4, ACACB, LIPC APP 698/4885ESR1 2003/4885ESR2 943/4885
US-20090304825-A1 ESTROGENIC EXTRACTS FOR USE IN TREATING VAGINAL AND VULVAR ATROPHY CYP19A1, SHBG, ESR1 APP 2398/4885ESR1 3/4885ESR2 7/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.