SCHEMBL7772085

SCHEMBL7772085

C=CCCNCC=CCOc1ccc(C(=O)C=CC=C(C)C)cc1F

nearest known ligand 0.34

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 3/20 0.34
ALDH1A1 P00352 1/20 0.34
PTPN1 P18031 3/20 0.32
POLB P06746 1/20 0.32
MAPT P10636 2/20 0.31
CYP3A4 P08684 1/20 0.31
BTK Q06187 2/20 0.31
EGFR P00533 1/20 0.31
LMNA P02545 1/20 0.31
BRD4 O60885 1/20 0.31
TUBB1 Q9H4B7 1/20 0.30
ABCB1 P08183 1/20 0.30
NPC1 O15118 1/20 0.30
RAB9A P51151 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7769135 0.90 PTGES (0.36) KDM4EALDH1A1PTPN1
SCHEMBL7768082 0.84 NPC1 (0.38) KDM4EALDH1A1PTPN1POLBMAPT
SCHEMBL7764172 0.83 KDM4E (0.33) KDM4EALDH1A1LMNANPC1RAB9A
SCHEMBL7764135 0.81 MAOB (0.36) ALDH1A1PTPN1MAPTLMNA
SCHEMBL7681554 0.81 LSS (0.46) KDM4EPTPN1MAPTLMNA
SCHEMBL7681546 0.81 LSS (0.46) KDM4EPTPN1MAPTLMNA
SCHEMBL7772100 0.80 KDM4E (0.33) KDM4EPTPN1POLBBTKEGFR
SCHEMBL7769445 0.80 KDM4E (0.36) KDM4EPOLBBRD4
SCHEMBL8047273 0.79 IL2 (0.35) KDM4EALDH1A1BRD4
Fumaric Acid SCHEMBL7681356 0.79 LSS (0.44) ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0778264-B1 Tertiary amines having antimycotic and cholesterol lowering activity HOFFMANN LA ROCHE (CH) 2001-07-11 EP claimed