SCHEMBL7772503

SCHEMBL7772503

CSc1ccc(C(O)(C[C@@H](C)C(N)(Oc2ccccc2)C(C)O)c2ccc(SC)cc2)cc1

nearest known ligand 0.39

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
KIF11 P52732 5/20 0.39
EDNRB P24530 2/20 0.35
EDNRA P25101 2/20 0.35
KDM4E B2RXH2 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.31
ALDH1A1 P00352 2/20 0.31
CYP2D6 P10635 1/20 0.31
CYP2C19 P33261 1/20 0.31
HSD17B10 Q99714 1/20 0.31
LMNA P02545 1/20 0.31
GRIN1 Q05586 4/20 0.30
GRIN2A Q12879 4/20 0.30
GRIN2D O15399 3/20 0.30
GRIN2C Q14957 3/20 0.30
GRIN2B Q13224 2/20 0.30
SLC6A4 P31645 2/20 0.30
MAOA P21397 1/20 0.30
SLC6A2 P23975 1/20 0.30
SLC6A3 Q01959 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7772520 0.86 KIF11 (0.43) KIF11SMN1; SMN2ALDH1A1CYP2D6CYP2C19
SCHEMBL7764655 0.85 KIF11 (0.45) KIF11SMN1; SMN2LMNA
SCHEMBL7764620 0.80 KIF11 (0.40) KIF11EDNRBEDNRAKDM4EALDH1A1
SCHEMBL7770270 0.80 KIF11 (0.41) KIF11
SCHEMBL7772500 0.72 LMNA (0.40) KIF11KDM4ECYP2D6LMNAMAOA
SCHEMBL6322832 0.69 ADRB2 (0.54) ALDH1A1CYP2D6SLC6A2
SCHEMBL6322160 0.69 SIGMAR1 (0.36) KIF11KDM4ESMN1; SMN2ALDH1A1CYP2D6
SCHEMBL6322829 0.69 ADRB2 (0.54) ALDH1A1CYP2D6SLC6A2
SCHEMBL6322158 0.69 SIGMAR1 (0.36) KIF11KDM4ESMN1; SMN2ALDH1A1CYP2D6
SCHEMBL11622889 0.68 KIF11 (0.47) KIF11SMN1; SMN2CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1107944-A1 AMINOALCOHOL DERIVATIVES AND THEIR USE AS BETA 3 ADRENERGIC AGONISTS FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 2001-06-20 EP disclosed
WO-2000012462-A1 AMINOALCOHOL DERIVATIVES AND THEIR USE AS BETA 3 ADRENERGIC AGONISTS FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 2000-03-09 WO disclosed