SCHEMBL7789908

SCHEMBL7789908

CCOC(=O)c1cc(NS(=O)(=O)c2ccc3ccccc3c2)ccc1Br

nearest known ligand 0.62

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HIF1A Q16665 1/20 0.62
MEN1 O00255 5/20 0.56
KMT2A Q03164 5/20 0.56
ALDH1A1 P00352 4/20 0.56
PKM P14618 2/20 0.55
PKLR P30613 1/20 0.55
AR P10275 1/20 0.55
PLAU P00749 2/20 0.54
SMN1; SMN2 Q16637 5/20 0.53
LMNA P02545 5/20 0.53
GAA P10253 2/20 0.53
HTT P42858 3/20 0.53
MAPT P10636 1/20 0.53
ATM Q13315 1/20 0.51
NHERF1 O14745 1/20 0.51
HDAC3 O15379 1/20 0.49
HDAC4 P56524 1/20 0.49
HDAC1 Q13547 1/20 0.49
HDAC7 Q8WUI4 1/20 0.49
HDAC2 Q92769 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7320847 0.89 PKM (0.64) HIF1AMEN1KMT2AALDH1A1PKM
SCHEMBL7791354 0.83 PLAU (0.72) HIF1AMEN1KMT2AALDH1A1PKM
SCHEMBL7789916 0.83 KMT2A (0.75) MEN1KMT2AALDH1A1PKMPKLR
SCHEMBL7319886 0.81 LMNA (0.69) HIF1AMEN1KMT2AALDH1A1PKM
SCHEMBL1883726 0.79 MEN1 (0.64) HIF1AMEN1KMT2AALDH1A1PKM
SCHEMBL6078420 0.78 PLAU (0.50) MEN1KMT2AALDH1A1PLAUSMN1; SMN2
SCHEMBL2894678 0.77 NHERF1 (0.71) HIF1AMEN1KMT2AALDH1A1SMN1; SMN2
SCHEMBL27939522 0.77 HIF1A (0.55) HIF1AMEN1KMT2AALDH1A1SMN1; SMN2
SCHEMBL26603234 0.76 HIF1A (0.96) HIF1ASMN1; SMN2LMNA
SCHEMBL2824645 0.76 AR (0.67) HIF1AMEN1KMT2AALDH1A1AR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6251917-B1 Benzamidoaldehydes and their use as cysteine protease inhibitors BASF AKTIENGESELLSCHAFT (DE) 2001-06-26 US disclosed