SCHEMBL7790169

SCHEMBL7790169

COc1ccc(S(=O)(=O)NC(CC(=O)O)c2cccc(NS(=O)(=O)c3cccc(NC(=N)N)c3)c2)cc1

nearest known ligand 0.51

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
ITGB3 P05106 3/20 0.49
ITGAV P06756 3/20 0.49
MAPT P10636 5/20 0.48
ALDH1A1 P00352 2/20 0.48
LMNA P02545 2/20 0.48
CYP19A1 P11511 1/20 0.47
ATM Q13315 1/20 0.47
KMT2A Q03164 2/20 0.47
SMN1; SMN2 Q16637 2/20 0.47
F2 P00734 1/20 0.46
TCF4 P15884 1/20 0.46
CTNNB1 P35222 1/20 0.46
MEN1 O00255 1/20 0.45
NPSR1 Q6W5P4 1/20 0.45
THRB P10828 1/20 0.45
HTT P42858 1/20 0.45
GAA P10253 1/20 0.44
HSD17B10 Q99714 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7786198 0.89 ITGB3 (0.49) ITGB3ITGAVMAPTALDH1A1LMNA
SCHEMBL7785662 0.88 MAPT (0.48) ITGB3MAPTALDH1A1LMNAATM
SCHEMBL7785637 0.87 ATM (0.50) ITGB3ITGAVMAPTALDH1A1ATM
SCHEMBL6366667 0.87 ITGB3 (0.60) ITGB3ITGAVALDH1A1ATM
SCHEMBL7781109 0.85 ITGB3 (0.49) ITGB3ITGAVALDH1A1ATMKMT2A
SCHEMBL7785592 0.85 ITGB3 (0.49) ITGB3ITGAVMAPTALDH1A1LMNA
SCHEMBL7785609 0.85 LMNA (0.45) ITGB3MAPTALDH1A1LMNAKMT2A
SCHEMBL7187012 0.83 MAPT (0.47) ITGB3ITGAVMAPTALDH1A1LMNA
SCHEMBL7786249 0.83 EEF2K (0.50) ITGB3ITGAVMAPTLMNAKMT2A
SCHEMBL13715863 0.82 PKM (0.46) ITGB3ITGAVMAPTALDH1A1LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1147079-A2 BETA-PHENYLALANINE DERIVATIVES AS INTEGRIN ANTAGONISTS Bayer Aktiengesellschaft (DE) 2001-10-24 EP disclosed
WO-2000041469-A2 β-PHENYLALANINE DERIVATIVES AS INTEGRIN ANTAGONISTS BAYER AKTIENGESELLSCHAFT (DE) 2000-07-20 WO disclosed