SCHEMBL7794250

SCHEMBL7794250

COc1cc(C=C(C(=O)OC(C)C)P(=O)(OC)OC)cc(OC)c1O

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTP4A3 O75365 2/20 0.51
PTP4A2 Q12974 2/20 0.51
PTP4A1 Q93096 2/20 0.51
CYP3A4 P08684 3/20 0.42
CYP1A2 P05177 2/20 0.42
CYP2C9 P11712 2/20 0.42
CYP2B6 P20813 2/20 0.42
CYP2D6 P10635 1/20 0.42
KMT2A Q03164 7/20 0.42
MAPT P10636 4/20 0.42
GAA P10253 2/20 0.42
PKM P14618 2/20 0.41
PTGS1 P23219 1/20 0.41
PTGS2 P35354 1/20 0.41
MEN1 O00255 4/20 0.40
ALDH1A1 P00352 2/20 0.40
ALOX5 P09917 2/20 0.38
ABL1 P00519 1/20 0.37
BCR P11274 1/20 0.37
LMNA P02545 3/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8842877 1.00 PTP4A3 (0.51) PTP4A3PTP4A2PTP4A1CYP3A4CYP1A2
SCHEMBL7793570 0.86 MAPT (0.51) CYP3A4CYP1A2CYP2C9CYP2B6CYP2D6
SCHEMBL8842889 0.84 ALDH1A1 (0.47) CYP1A2KMT2AMAPTMEN1ALDH1A1
SCHEMBL7784722 0.84 ALDH1A1 (0.47) CYP1A2KMT2AMAPTMEN1ALDH1A1
SCHEMBL8842926 0.81 GAA (0.44) CYP1A2MAPTGAAALDH1A1KDM4E
SCHEMBL7784710 0.81 GAA (0.44) CYP1A2MAPTGAAALDH1A1KDM4E
SCHEMBL2903666 0.80 PTP4A3 (0.57) PTP4A3PTP4A2PTP4A1CYP3A4CYP1A2
SCHEMBL7790430 0.78 POLB (0.53) KMT2AMAPTMEN1ALDH1A1KDM4E
SCHEMBL7784713 0.78 HDAC1 (0.48) KMT2AMAPTALDH1A1LMNAHPGD
SCHEMBL7784715 0.78 HDAC1 (0.48) KMT2AMAPTALDH1A1LMNAHPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0723969-B1 Phosphonocarboxylic acid derivatives and their use in treating degenerative articular ailments HOECHST AG (DE) 2001-11-14 EP disclosed
US-5627173-A Phosphonoacetic acid derivatives and their use for treating degenerative joint disorders HOECHST AKTIENGESELLSCHAFT (DE) 1997-05-06 US disclosed
EP-0723969-A1 Phosphonocarboxylic acid derivatives and their use in treating degenerative articular ailments HOECHST AKTIENGESELLSCHAFT (DE) 1996-07-31 EP disclosed