SCHEMBL7798387

SCHEMBL7798387

O=[P](c1cc(C(F)(F)F)cc(C(F)(F)F)c1)c1cc(C(F)(F)F)cc(C(F)(F)F)c1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CES2 O00748 1/20 0.46
IDO1 P14902 2/20 0.37
RXRA P19793 2/20 0.36
RXRB P28702 2/20 0.36
RXRG P48443 2/20 0.36
MAPT P10636 1/20 0.36
ALDH1A1 P00352 1/20 0.34
CYP3A4 P08684 1/20 0.34
HPGD P15428 1/20 0.34
ALOX15 P16050 1/20 0.34
TSHR P16473 1/20 0.34
HIF1A Q16665 1/20 0.34
TXNRD1 Q16881 1/20 0.34
TXNRD3 Q86VQ6 1/20 0.34
TXNRD2 Q9NNW7 1/20 0.34
TDP1 Q9NUW8 1/20 0.34
XPO1 O14980 1/20 0.34
LMNA P02545 1/20 0.33
GPR35 Q9HC97 1/20 0.33
P2RX1 P51575 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL383565 0.78 CES2 (0.44) CES2IDO1RXRARXRBRXRG
SCHEMBL7795645 0.77 CES2 (0.48) CES2IDO1MAPTALDH1A1TSHR
SCHEMBL440959 0.76 CES2 (0.58) CES2IDO1RXRARXRBRXRG
SCHEMBL16861287 0.76 CES2 (0.42) CES2IDO1RXRARXRBRXRG
SCHEMBL15329899 0.76 CES2 (0.42) CES2IDO1RXRARXRBRXRG
SCHEMBL2879502 0.74 CES2 (0.41) CES2IDO1RXRARXRBRXRG
SCHEMBL497733 0.74 CES2 (0.41) CES2IDO1RXRARXRBRXRG
SCHEMBL2227681 0.74 CES2 (0.41) CES2IDO1RXRARXRBRXRG
SCHEMBL7526444 0.74 CES2 (0.46) CES2ALDH1A1TSHR
SCHEMBL1305235 0.74 GABRA1 (0.46) RXRARXRBRXRGMAPTALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-10072033-B2 N-(phosphinoalkyl)-N-(thioalkyl)amine derivative, method for producing same, and metal complex thereof TAKASAGO INTERNATIONAL CORPORATION (JP) 2018-09-11 US disclosed
US-20170233418-A1 N-(PHOSPHINOALKYL)-N-(THIOALKYL)AMINE DERIVATIVE, METHOD FOR PRODUCING SAME, AND METAL COMPLEX THEREOF TAKASAGO INTERNATIONAL CORPORATION (JP) 2017-08-17 US disclosed
EP-0731105-B1 Optically active tertiary phosphine compounds, transition metal complexes comprising the same as ligands and process for preparing optically active organic silicon compounds using said transition metal complexes SUMITOMO CHEMICAL CO (JP) 2001-12-05 EP disclosed
US-5621129-A Optically active tertiary phosphine compound, transition metal complex comprising the same as ligand and process for preparing optically active organic silicon compound using said transition metal complex SUMITOMO CHEMICAL CO., LTD. (JP) 1997-04-15 US disclosed
EP-0731105-A1 Optically active tertiary phosphine compounds, transition metal complexes comprising the same as ligands and process for preparing optically active organic silicon compounds using said transition metal complexes SUMITOMO CHEMICAL COMPANY LIMITED (JP) 1996-09-11 EP disclosed
US-5484902-A HYDROCYANATION OF VINYL AROMATICS E. I. DU PONT DE NEMOURS AND COMPANY (US) 1996-01-16 US disclosed
US-5312957-A 2-/6-Methoxy-2-naphthalene/propionitrile E. I. DU PONT DE NEMOURS AND COMPANY (US) 1994-05-17 US disclosed
US-5175335-A Reacting vinyl aryl compounds with a source of hydrocyanic acid in presence of nickle zero valent compound and nonracemic bidentate organophosphorus ligand E. I. DU PONT DE NEMOURS AND COMPANY (US) 1992-12-29 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20170233418-A1 N-(PHOSPHINOALKYL)-N-(THIOALKYL)AMINE DERIVATIVE, METHOD FOR PRODUCING SAME, AND METAL COMPLEX THEREOF NSFL1C, TST, NCL CES2 2520/4885IDO1 2171/4885RXRA 4650/4885
US-10072033-B2 N-(phosphinoalkyl)-N-(thioalkyl)amine derivative, method for producing same, and metal complex thereof NSFL1C, TST, NCL CES2 2520/4885IDO1 2171/4885RXRA 4650/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.