SCHEMBL7798437

SCHEMBL7798437

NCCc1ccc(Oc2ccccc2)cc1.O=C(O)c1ccc(-c2ccccc2)cc1.O=Cc1cc(C(F)(F)F)cc(C(F)(F)F)c1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SRD5A2 P31213 3/20 0.47
RXRA P19793 1/20 0.45
RXRB P28702 1/20 0.45
RXRG P48443 1/20 0.45
MAPK14 Q16539 2/20 0.44
MAOB P27338 2/20 0.44
MEN1 O00255 1/20 0.42
KMT2A Q03164 1/20 0.42
LTA4H P09960 1/20 0.42
EPHX2 P34913 1/20 0.42
TRIM24 O15164 1/20 0.41
TRIM33 Q9UPN9 1/20 0.41
PTPN2 P17706 2/20 0.41
PTPN1 P18031 2/20 0.41
ACP1 P24666 2/20 0.41
NR4A2 P43354 1/20 0.40
PTGES O14684 1/20 0.40
ALOX5 P09917 1/20 0.40
LPAR1 Q92633 1/20 0.39
LPAR5 Q9H1C0 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Benzoic Acid SCHEMBL7801470 0.94 SRD5A2 (0.48) SRD5A2MAPK14MAOBMEN1KMT2A
SCHEMBL8035858 0.91 MAOB (0.46) RXRARXRBRXRGMAOBTRIM24
4-Methylbenzoic Acid SCHEMBL7802556 0.91 SRD5A2 (0.46) SRD5A2MAPK14MEN1KMT2ALTA4H
SCHEMBL7798600 0.91 SRD5A2 (0.46) SRD5A2RXRARXRBMAPK14MEN1
Phenethylamine SCHEMBL7799179 0.91 RXRA (0.52) SRD5A2RXRARXRBRXRGMAOB
SCHEMBL7802496 0.90 RXRA (0.46) RXRARXRBRXRGMAOBTRIM24
Tyramine SCHEMBL8035895 0.89 RXRA (0.48) SRD5A2RXRARXRBRXRGMAOB
SCHEMBL7798406 0.89 MAOB (0.46) MAPK14MAOBMEN1KMT2ALTA4H
SCHEMBL7802656 0.88 RXRA (0.47) SRD5A2RXRARXRBRXRGMAOB
SCHEMBL8035116 0.86 PTGES (0.48) RXRARXRBRXRGMAOBMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1076649-A1 ISOQUINOLINE COMPOUND MELANOCORTIN RECEPTOR LIGANDS AND METHODS OF USING SAME TREGA BIOSCIENCES, INC. (US) 2001-02-21 EP disclosed
US-6127381-A A MELANOCORTIN RECEPTOR LIGAND FOR REGULATING FOOD INTAKE AND BODY WEIGHT, REGULATING CYTOKINE ACTIVITY, ANTI-INFLAMMATORY ACTIVITY LION BIOSCIENCE AG (DE) 2000-10-03 US disclosed
WO-1999055679-A1 ISOQUINOLINE COMPOUND MELANOCORTIN RECEPTOR LIGANDS AND METHODS OF USING SAME TREGA BIOSCIENCES, INC. (US) 1999-11-04 WO disclosed