SCHEMBL7804752

SCHEMBL7804752

CC(C)(C)OC(=O)N1C[C@H](O[Si](C)(C)C(C)(C)C)C[C@H]1C(O)C1CCN(C(=O)OCc2ccc([N+](=O)[O-])cc2)CC1

nearest known ligand 0.39

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.39
MAPT P10636 3/20 0.39
LMNA P02545 2/20 0.39
GPR119 Q8TDV5 2/20 0.36
SMN1; SMN2 Q16637 1/20 0.35
HPGD P15428 1/20 0.35
PARP1 P09874 1/20 0.35
CCR5 P51681 2/20 0.35
MCL1 Q07820 5/20 0.34
KDM4E B2RXH2 1/20 0.34
NR1D1 P20393 1/20 0.34
KMT2A Q03164 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7804783 0.93 ALDH1A1 (0.38) ALDH1A1MAPTLMNAGPR119HPGD
SCHEMBL9399096 0.83 ALDH1A1 (0.43) ALDH1A1MAPTLMNAGPR119HPGD
SCHEMBL9399315 0.82 ALDH1A1 (0.42) ALDH1A1MAPTLMNAGPR119HPGD
SCHEMBL9020556 0.81 CCR5 (0.43) ALDH1A1MAPTLMNAGPR119HPGD
SCHEMBL8098546 0.80 MCL1 (0.36) ALDH1A1MAPTLMNAGPR119HPGD
SCHEMBL7805751 0.79 SMN1; SMN2 (0.41) ALDH1A1MAPTLMNASMN1; SMN2KDM4E
SCHEMBL7804672 0.78 SMN1; SMN2 (0.40) ALDH1A1MAPTLMNASMN1; SMN2HPGD
SCHEMBL9520871 0.78 CCR5 (0.36) ALDH1A1MAPTLMNASMN1; SMN2HPGD
SCHEMBL7809902 0.78 PRMT5 (0.36) GPR119HPGD
SCHEMBL7806059 0.78 PRMT5 (0.36) GPR119HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0773222-B1 CARBAPENEM DERIVATIVE EISAI CO LTD (JP) 2001-10-04 EP disclosed
US-6037341-A HAVING POTENT ANTIMICROBIAL EFFECTS OVER GRAM-POSITIVE BACTERIA AND GRAM-NEGATIVE BACTERIA EISAI CO., LTD. (JP) 2000-03-14 US disclosed
EP-0773222-A1 NOVEL CARBAPENEM DERIVATIVE Eisai Co., Ltd. (JP) 1997-05-14 EP disclosed