SCHEMBL7811209

SCHEMBL7811209

Cc1cnc2c3c(nccc13)C(=O)c1ccccc1-2

nearest known ligand 0.53

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
MAOA P21397 3/20 0.53
ALDH1A1 P00352 1/20 0.50
KMT2A Q03164 1/20 0.46
PTPRC P08575 2/20 0.45
CTSL P07711 1/20 0.45
CTSS P25774 1/20 0.45
PTPN13 Q12923 1/20 0.45
TOP2A P11388 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7804497 0.82 MAOA (0.53) MAOAALDH1A1KMT2APTPRCCTSL
SCHEMBL7813560 0.82 MAOA (0.53) MAOAALDH1A1KMT2APTPRCCTSL
SCHEMBL7811692 0.82 MAOA (0.53) MAOAALDH1A1KMT2APTPRCCTSL
SCHEMBL7804334 0.81 MAOA (0.53) MAOAALDH1A1KMT2A
Sampangine SCHEMBL6230423 0.75 MAOA (0.74) MAOAALDH1A1KMT2APTPRCCTSL
Benzosampangine SCHEMBL20259217 0.73 TOP2A (0.79) MAOAALDH1A1PTPRCCTSLCTSS
Benzosampangine SCHEMBL29601408 0.73 TOP2A (0.79) MAOAALDH1A1PTPRCCTSLCTSS
SCHEMBL28154272 0.72 BRCA1 (0.46) MAOA
SCHEMBL23235907 0.70 ALDH1A1 (0.55) MAOAALDH1A1KMT2APTPRCCTSL
Cleistopholine SCHEMBL6358965 0.70 ALDH1A1 (0.55) MAOAALDH1A1KMT2APTPRCCTSL

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0588796-B1 SAMPANGINE DERIVATIVES USEFUL AS ANTIFUNGAL AND ANTIMYCOBACTERIAL AGENTS UNIV MISSISSIPPI (US) 2001-04-04 EP disclosed
US-5530004-A ADMINISTERING SAMPANGINE AND CLEISTOPHOLINE ANALOGS THE UNIVERSITY OF MISSISSIPPI (US) 1996-06-25 US disclosed
EP-0588796-A1 NEW COMPOUNDS AND COMPOSITIONS USEFUL AS ANTIFUNGAL AND ANTIMYCOBACTERIAL AGENTS THE UNIVERSITY OF MISSISSIPPI (US) 1994-03-30 EP disclosed
US-5227383-A Sampangine analogs THE UNIVERSITY OF MISSISSIPPI (US) 1993-07-13 US disclosed
WO-1992022297-A1 NEW COMPOUNDS AND COMPOSITIONS USEFUL AS ANTIFUNGAL AND ANTIMYCOBACTERIAL AGENTS THE UNIVERSITY OF MISSISSIPPI (US) 1992-12-23 WO disclosed