SCHEMBL7811405

SCHEMBL7811405

COc1ccc(F)c2c1C(=O)c1nccnc1C2=O

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 5/20 0.46
KDM4E B2RXH2 5/20 0.46
MAPK1 P28482 4/20 0.46
HTT P42858 3/20 0.46
RAB9A P51151 2/20 0.46
NPSR1 Q6W5P4 2/20 0.46
S1PR4 O95977 1/20 0.46
HSP90AA1 P07900 1/20 0.46
G6PD P11413 1/20 0.46
S1PR1 P21453 1/20 0.46
OPRK1 P41145 1/20 0.46
CACNA1B Q00975 1/20 0.46
APBA1 Q02410 1/20 0.46
MCL1 Q07820 1/20 0.46
APOBEC3G Q9HC16 1/20 0.46
TLR9 Q9NR96 1/20 0.46
USP8 P40818 2/20 0.45
USP7 Q93009 2/20 0.45
ALDH1A1 P00352 5/20 0.44
KMT2A Q03164 4/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7817043 0.84 ALDH1A1 (0.45) USP8USP7ALDH1A1KMT2AMEN1
SCHEMBL7810488 0.75 MAPT (0.51) MAPTKDM4EMAPK1HTTRAB9A
SCHEMBL7810480 0.75 MAPT (0.51) MAPTKDM4EMAPK1HTTRAB9A
SCHEMBL7809872 0.74 MEN1 (0.39) MAPTKDM4EMAPK1RAB9ANPSR1
SCHEMBL7823380 0.74 ALDH1A1 (0.37) ALDH1A1KMT2AMEN1TDP1THRB
SCHEMBL11134106 0.71 MAPT (0.73) MAPTKDM4EMAPK1HTTRAB9A
SCHEMBL8996375 0.69 TOP1 (0.52) MAPTKDM4EMAPK1HTTRAB9A
SCHEMBL6407586 0.68 MAPT (0.40) MAPTKDM4EMAPK1HTTRAB9A
SCHEMBL7809098 0.67 TDP2 (0.59) KMT2AMEN1TDP1THRBHKDC1
SCHEMBL6407178 0.66 MAPT (0.50) MAPTKDM4EMAPK1HTTRAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0750619-B1 HETERO-ANNULATED INDAZOLES NOVUSPHARMA SPA (IT) 2001-05-30 EP disclosed
US-5596097-A ANTITUMOR AGENTS THE UNIVERSITY OF VERMONT (US) 1997-01-21 US disclosed
EP-0750619-A1 HETERO-ANNULATED INDAZOLES BOEHRINGER MANNHEIM ITALIA S.p.A. (IT) 1997-01-02 EP disclosed
WO-1995024407-A1 HETERO-ANNULATED INDAZOLES BOEHRINGER MANNHEIM ITALIA, S.P.A. (IT) 1995-09-14 WO disclosed