N-Desmethylclozapine

N-Desmethylclozapine

SCHEMBL781423

Clc1ccc2c(c1)N=C(N1CCNCC1)c1ccccc1N2

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Full drug profile on Sugi Atlas →

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DRD2 P14416 17/20 1.00
DRD1 P21728 9/20 1.00
CHRM1 P11229 5/20 1.00
CYP1A2 P05177 3/20 1.00
CHRM2 P08172 3/20 1.00
CHRM4 P08173 3/20 1.00
CYP3A4 P08684 3/20 1.00
CHRM5 P08912 3/20 1.00
CYP2D6 P10635 3/20 1.00
CHRM3 P20309 3/20 1.00
KCNH2 Q12809 3/20 1.00
MTOR P42345 2/20 1.00
DRD3 P35462 4/20 0.76
DRD4 P21917 3/20 0.76
DRD5 P21918 3/20 0.76
HRH1 P35367 3/20 0.76
HRH4 Q9H3N8 2/20 0.76
MEN1 O00255 2/20 0.76
LMNA P02545 2/20 0.76
ADRB2 P07550 2/20 0.76

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
N-Desmethylclozapine SCHEMBL29365906 1.00 DRD2 (1.00) DRD2DRD1CHRM1CYP1A2CHRM2
N-Desmethylclozapine SCHEMBL29360816 1.00 DRD2 (1.00) DRD2DRD1CHRM1CYP1A2CHRM2
N-Desmethylclozapine SCHEMBL30416482 1.00 DRD2 (1.00) DRD2DRD1CHRM1CYP1A2CHRM2
SCHEMBL3431059 0.95 DRD2 (0.91) DRD2DRD1CHRM1CYP1A2CHRM2
SCHEMBL20887469 0.92 DRD2 (0.88) DRD2DRD1CHRM1CYP1A2CHRM2
SCHEMBL3411298 0.91 DRD2 (0.83) DRD2DRD1CHRM1CYP1A2CHRM2
SCHEMBL3408005 0.90 DRD2 (0.82) DRD2DRD1CHRM1CYP1A2CHRM2
SCHEMBL3411946 0.90 DRD2 (0.82) DRD2DRD1CHRM1CYP1A2CHRM2
SCHEMBL3407780 0.90 DRD2 (0.81) DRD2DRD1CHRM1CYP1A2CHRM2
SCHEMBL3411880 0.89 DRD2 (0.80) DRD2DRD1CHRM1CYP1A2CHRM2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 365 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20230288372-A1 Systems and Methods for Separating Compounds of Similar Mass by Differential Mobility Spectrometry DH TECHNOLOGIES DEVELOPMENT PTE. LTD. (SG) 2023-09-14 US claimed
EP-4100733-A1 SYSTEMS AND METHODS FOR SEPARATING COMPOUNDS OF SIMILAR MASS BY DIFFERENTIAL MOBILITY SPECTROMETRY DH Technologies Development Pte. Ltd. (SG) 2022-12-14 EP claimed
WO-2021156775-A1 SYSTEMS AND METHODS FOR SEPARATING COMPOUNDS OF SIMILAR MASS BY DIFFERENTIAL MOBILITY SPECTROMETRY DH TECHNOLOGIES DEVELOPMENT PTE. LTD. (SG) 2021-08-12 WO claimed
US-20200289489-A1 COMBINATION FOR TREATING PAIN REGENTS OF THE UNIVERSITY OF MINNESOTA (US) 2020-09-17 US claimed
EP-3432884-A1 COMBINATION FOR TREATING PAIN Regents of the University of Minnesota (US) 2019-01-30 EP claimed
WO-2017165558-A1 COMBINATION FOR TREATING PAIN REGENTS OF THE UNIVERSITY OF MINNESOTA (US) 2017-09-28 WO claimed
EP-3137658-A1 USE OF KNOWN COMPOUNDS AS D-AMINO ACID OXIDASE INHIBITORS Tseng, Yufeng, Jane (US) 2017-03-08 EP claimed
WO-2016023997-A1 HETEROCYCLIC COMPOUNDS WITH WORKING MEMORY ENHANCING ACTIVITY RED BULL GMBH (AT) 2016-02-18 WO claimed
US-20150374712-A1 Combinations of Dopamine D2 Receptor Blockade With Norepinephrine Reuptake Inhibition and with Norepinephrine Alpha 2 Receptor Blockade GREEN ALAN I (US) 2015-12-31 US claimed
WO-2012161938-A1 CLOZAPINE IMMUNOASSAY SALADAX BIOMEDICAL INC. (US) 2012-11-29 WO claimed
WO-2006001866-A2 CRYSTALLINE FORMS OF N-DESMETHYLCLOZAPINE ACADIA PHARMACEUTICALS INC. (US) 2006-01-05 WO claimed
EP-1596867-A2 TREATMENT OF PSYCHOSIS WITH A MUSCARINIC M1 RECEPTOR ECTOPIC ACTIVATOR Merck & Co., Inc. (US) 2005-11-23 EP claimed
EP-1589974-A2 USE OF N-DESMETHYLCLOZAPINE TO TREAT HUMAN NEUROPSYCHIATRIC DISEASE Acadia Pharmaceuticals Inc. (US) 2005-11-02 EP claimed
EP-1587789-A2 SELECTIVE SEROTONIN 2A/2C RECEPTOR INVERSE AGONISTS AS THERAPEUTICS FOR NEURODEGENERATIVE DISEASES Acadia Pharmaceuticals Inc. (US) 2005-10-26 EP claimed
WO-2005063254-A2 AMINO SUBSTITUTED DIARYL[A,D]CYCLOHEPTENE ANALOGS AS MUSCARINIC AGONISTS AND METHODS OF TREATMENT OF NEUROPSYCHIATRIC DISORDERS ACADIA PHARMACEUTICALS INC. (US) 2005-07-14 WO claimed
US-20050080084-A1 Compositions of a cyclooxygenase-2 selective inhibitor and a serotonin-modulating agent for the treatment of central nervous system damage PHARMACIA CORPORATION 2005-04-14 US claimed
WO-2005018541-A2 COX-2 INHIBITOR AND SEROTONIN MODULATOR FOR TREATING CNS DAMAGE PHARMACIA CORPORATION (US) 2005-03-03 WO claimed
WO-2004073639-A2 TREATMENT OF PSYCHOSIS WITH A MUSCARINIC M1 RECEPTOR ECTOPIC ACTIVATOR MERCK & CO. INC. (US) 2004-09-02 WO claimed
WO-2004064753-A2 USE OF N-DESMETHYLCLOZAPINE TO TREAT HUMAN NEUROPSYCHIATRIC DISEASE ACADIA PHARMACEUTICALS INC (US) 2004-08-05 WO claimed
WO-2004064738-A2 SELECTIVE SEROTONIN 2A/2C RECEPTOR INVERSE AGONISTS AS THERAPEUTICS FOR NEURODEGENERATIVE DISEASES ACADIA PHARMACEUTICALS INC. (US) 2004-08-05 WO claimed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20050080084-A1 Compositions of a cyclooxygenase-2 selective inhibitor and a serotonin-modulating agent for the treatment of central nervous system damage TPH2, TPH1, HTR2A DRD2 327/4885DRD1 1384/4885CHRM1 962/4885
US-20200289489-A1 COMBINATION FOR TREATING PAIN OPRL1, ACHE, OPRK1 DRD2 1728/4885DRD1 3062/4885CHRM1 915/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.