SCHEMBL7827339

SCHEMBL7827339

COc1cc2c(cc1OC)CC1(CC2)NC(=O)CN(C)C1=O

nearest known ligand 0.42

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
GAA P10253 1/20 0.42
SMN1; SMN2 Q16637 1/20 0.42
MAOA P21397 2/20 0.39
MAOB P27338 2/20 0.39
SLC6A4 P31645 1/20 0.39
MEN1 O00255 1/20 0.39
KMT2A Q03164 1/20 0.39
ALDH1A1 P00352 3/20 0.39
LMNA P02545 1/20 0.39
MAPT P10636 1/20 0.39
HTT P42858 1/20 0.39
PDE4D Q08499 1/20 0.36
BRD4 O60885 2/20 0.36
CA7 P43166 1/20 0.35
SRC P12931 1/20 0.34
ABCB1 P08183 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8841801 0.79 ALDH1A1 (0.53) SMN1; SMN2MEN1KMT2AALDH1A1LMNA
SCHEMBL7822652 0.75 ACHE (0.41) GAASMN1; SMN2MAOAALDH1A1PDE4D
SCHEMBL11073395 0.71 GAA (0.39) GAASMN1; SMN2MAOAMAOBSLC6A4
SCHEMBL7815545 0.66 ALDH1A1 (0.40) GAASMN1; SMN2MAOAALDH1A1ABCB1
SCHEMBL30340281 0.62 CYP19A1 (0.48) GAAKMT2AMAPTSRC
SCHEMBL7429093 0.62 CYP19A1 (0.48) GAAKMT2AMAPTSRC
SCHEMBL16339494 0.62 CYP11B1 (0.57) GAASLC6A4KMT2AALDH1A1MAPT
SCHEMBL1814392 0.61 BACE1 (0.51) ALDH1A1LMNAMAPTHTTBRD4
SCHEMBL28447344 0.61 HTR5A (0.42) MEN1KMT2ALMNAMAPT
SCHEMBL7830514 0.60 MAOA (0.44) GAASMN1; SMN2MAOAMAOBSLC6A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0712845-B1 Amine compounds, their production and use TAKEDA CHEMICAL INDUSTRIES LTD (JP) 2001-10-17 EP disclosed
US-5633248-A GONADOTROPIN-RELEASING HORMONE RECEPTOR ANTAGONISTS, DIARYLALKYLIDENEDIAMINES TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1997-05-27 US disclosed
US-5591849-A TREATMENT OF CENTRAL NERVOUS SYSTEM DISORDERS, INHIBITORS OF AMINE, AMINE OXIDASE B, AND CALCIUM ION UPTAKE, NEUROPATHY, DYSMNESIA TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1997-01-07 US disclosed
EP-0712845-A1 Amine compounds, their production and use TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1996-05-22 EP disclosed
EP-0670313-A1 Spiro compounds, their production and use TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1995-09-06 EP disclosed