SCHEMBL7823112

SCHEMBL7823112

CCCC(CCC)Nc1nc(C)nc(Oc2c(Br)cc(C(C)(C)O)cc2OC)c1[N+](=O)[O-]

nearest known ligand 0.36

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
CRHR1 P34998 5/20 0.36
EDNRB P24530 1/20 0.32
EDNRA P25101 1/20 0.32
MAPK1 P28482 2/20 0.31
ALDH1A1 P00352 1/20 0.31
MAPT P10636 1/20 0.31
LMNA P02545 1/20 0.30
GAA P10253 1/20 0.30
SMN1; SMN2 Q16637 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7820028 0.88 CRHR1 (0.34) CRHR1EDNRBEDNRAMAPK1ALDH1A1
SCHEMBL7827120 0.85 TLR7 (0.35) CRHR1
SCHEMBL7820032 0.80 CRHR1 (0.35) CRHR1EDNRBEDNRAMAPK1ALDH1A1
SCHEMBL6894855 0.70
SCHEMBL7944720 0.70 CRHR1 (0.34) CRHR1
SCHEMBL5844675 0.68 CRHR1 (0.50) CRHR1
SCHEMBL5844265 0.66 CRHR1 (0.42) CRHR1
SCHEMBL6432632 0.65 ALDH1A1 (0.38) CRHR1MAPK1ALDH1A1MAPTLMNA
SCHEMBL7477014 0.65 KEAP1 (0.38) CRHR1ALDH1A1MAPTLMNA
SCHEMBL5844211 0.65 CRHR1 (0.38) CRHR1MAPK1ALDH1A1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0901476-A4 ARYLOXY- AND ARYLTHIO-FUSED PYRIDINES AND PYRIMIDINES AND DERIVATIVES DU PONT PHARM CO (US) 2001-08-16 EP disclosed
US-6258809-B1 NERVOUS SYSTEM DISORDERS, ANTIDEPRESSANTS AND PSYCHIATRY DUPONT PHARMACEUTICALS COMPANY 2001-07-10 US disclosed
US-6124300-A Aryloxy- and arylthio- fused pyridines and pyrimidines and derivatives DUPONT PHARMACEUTICALS (US) 2000-09-26 US disclosed
EP-0901476-A1 ARYLOXY- AND ARYLTHIO-FUSED PYRIDINES AND PYRIMIDINES AND DERIVATIVES Du Pont Pharmaceuticals Company (US) 1999-03-17 EP disclosed
WO-1997035846-A1 ARYLOXY- AND ARYLTHIO-FUSED PYRIDINES AND PYRIMIDINES AND DERIVATIVES DUPONT PHARMACEUTICALS COMPANY (US) 1997-10-02 WO disclosed