SCHEMBL7823769

SCHEMBL7823769

Cn1nnnc1Cc1ccc([N+](=O)[O-])cc1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
POLB P06746 1/20 0.49
ALDH1A1 P00352 6/20 0.45
NPC1 O15118 2/20 0.45
LMNA P02545 2/20 0.44
KCNJ1 P48048 1/20 0.43
KCNH2 Q12809 1/20 0.43
LOXL2 Q9Y4K0 1/20 0.42
MAPT P10636 3/20 0.42
RAB9A P51151 1/20 0.42
TGM2 P21980 1/20 0.42
HRH3 Q9Y5N1 1/20 0.41
PTK2 Q05397 1/20 0.41
CYP19A1 P11511 1/20 0.40
KMT2A Q03164 1/20 0.40
CA12 O43570 1/20 0.40
CA1 P00915 1/20 0.40
CA2 P00918 1/20 0.40
CA9 Q16790 1/20 0.40
CA14 Q9ULX7 1/20 0.40
TSHR P16473 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4825713 0.85 ALDH1A1 (0.49) POLBALDH1A1NPC1LMNALOXL2
SCHEMBL5654058 0.78 CYP1A2 (0.45) POLBALDH1A1NPC1LMNAMAPT
SCHEMBL27631985 0.78 ALDH1A1 (0.52) ALDH1A1LMNAMAPTCYP19A1KMT2A
SCHEMBL6358697 0.77 PKM (0.58) ALDH1A1LMNAMAPTSMN1; SMN2
SCHEMBL12414593 0.77 TRPV1 (0.66) ALDH1A1TGM2CYP2C19SMN1; SMN2
SCHEMBL4834216 0.76 ALDH1A1 (0.45) ALDH1A1NPC1LMNARAB9ACYP19A1
SCHEMBL3824667 0.76 ALDH1A1 (0.55) POLBALDH1A1LMNATSHRSMN1; SMN2
SCHEMBL4409003 0.75 CNR2 (0.49) ALDH1A1LMNAKMT2A
SCHEMBL1674067 0.73 PTGS2 (0.57) ALDH1A1LMNAMAPTRAB9AKMT2A
SCHEMBL7823805 0.72 HTR1A (0.41) ALDH1A1NPC1RAB9ASMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0630374-B1 IMIDAZOLE, TRIAZOLE AND TETRAZOLE DERIVATIVES MERCK SHARP & DOHME (GB) 2001-09-05 EP disclosed
US-5510362-A VASOCONSTRUCTION MERCK, SHARP AND DOHME LIMITED (GB) 1996-04-23 US disclosed
EP-0630374-A1 IMIDAZOLE, TRIAZOLE AND TETRAZOLE DERIVATIVES MERCK SHARP & DOHME LTD. (GB) 1994-12-28 EP disclosed
WO-1993018029-A1 IMIDAZOLE, TRIAZOLE AND TETRAZOLE DERIVATIVES MERCK SHARP & DOHME LIMITED (GB) 1993-09-16 WO disclosed