SCHEMBL7823967

SCHEMBL7823967

COc1ccc(C(CCCI)(CNC=O)c2ccccc2)cc1

nearest known ligand 0.43

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
KIF11 P52732 7/20 0.43
KCNH2 Q12809 1/20 0.43
LMNA P02545 4/20 0.39
SMN1; SMN2 Q16637 2/20 0.39
HTT P42858 1/20 0.39
CCR1 P32246 1/20 0.36
CCR3 P51677 1/20 0.36
DRD2 P14416 1/20 0.36
DRD4 P21917 1/20 0.36
DRD3 P35462 1/20 0.36
MEN1 O00255 2/20 0.36
KMT2A Q03164 2/20 0.36
ALDH1A1 P00352 4/20 0.35
KDM4E B2RXH2 3/20 0.35
MAPT P10636 2/20 0.35
TP53 P04637 1/20 0.35
F10 P00742 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7817328 0.88 ADH1B (0.38) KIF11MEN1KMT2AALDH1A1
SCHEMBL7824381 0.88 KIF11 (0.43) KIF11KCNH2LMNASMN1; SMN2HTT
SCHEMBL7827162 0.84 ADH1B (0.37) ALDH1A1
SCHEMBL7830286 0.83 KIF11 (0.39) KIF11LMNASMN1; SMN2HTTCCR1
SCHEMBL7466786 0.77 MCHR1 (0.54) LMNACCR1CCR3DRD2ALDH1A1
Hydrochloric Acid SCHEMBL7464242 0.76 MCHR1 (0.54) LMNACCR1CCR3DRD2ALDH1A1
SCHEMBL8894063 0.76 ADH1B (0.37) MEN1KMT2AALDH1A1
SCHEMBL7817246 0.76 ADH1B (0.37) MEN1KMT2AALDH1A1
SCHEMBL8892472 0.75 KIF11 (0.33) KIF11
SCHEMBL7462124 0.74 CCR1 (0.67) LMNACCR1CCR3MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0712845-B1 Amine compounds, their production and use TAKEDA CHEMICAL INDUSTRIES LTD (JP) 2001-10-17 EP disclosed
WO-1997024325-A1 DIPHENYLMETHANE DERIVATIVES AS MIP-1α/RANTES RECEPTOR ANTAGONISTS TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1997-07-10 WO disclosed
US-5633248-A GONADOTROPIN-RELEASING HORMONE RECEPTOR ANTAGONISTS, DIARYLALKYLIDENEDIAMINES TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1997-05-27 US disclosed
EP-0712845-A1 Amine compounds, their production and use TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1996-05-22 EP disclosed