SCHEMBL7833244

SCHEMBL7833244

CC(C)Oc1cc(CC(NC(=O)CNC(=O)c2cccc(NC=NN)c2)C(=O)O)cc(OC(C)C)c1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GPR139 Q6DWJ6 9/20 0.43
ITGB1 P05556 6/20 0.41
ITGB3 P05106 5/20 0.41
ITGAV P06756 5/20 0.41
ITGA2B P08514 3/20 0.41
ITGB5 P18084 3/20 0.41
GPR132 Q9UNW8 1/20 0.41
ITGA5 P08648 3/20 0.39
MDM2 Q00987 2/20 0.39
MDM4 O15151 1/20 0.39
NPC1 O15118 1/20 0.39
ALDH1A1 P00352 1/20 0.39
LMNA P02545 1/20 0.39
ALOX12 P18054 1/20 0.39
RAB9A P51151 1/20 0.39
SMN1; SMN2 Q16637 1/20 0.39
MEN1 O00255 1/20 0.39
KMT2A Q03164 1/20 0.39
ATM Q13315 1/20 0.39
F2 P00734 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6778010 0.91 GPR139 (0.49) GPR139GPR132ALDH1A1SMN1; SMN2MEN1
SCHEMBL7837425 0.91 GPR139 (0.40) GPR139ITGB1ITGB3ITGAVITGA5
SCHEMBL7823801 0.90 KMT2A (0.43) GPR139ITGB1ITGB3ITGAVITGA2B
SCHEMBL6778268 0.86 GPR139 (0.44) GPR139ITGB1ITGB3ITGAVITGA2B
SCHEMBL6775970 0.86 GPR132 (0.49) GPR139ITGB1ITGB3ITGAVITGA2B
SCHEMBL3051751 0.85 GPR139 (0.44) GPR139ITGB1ITGB3ITGAVITGB5
SCHEMBL6777818 0.85 ITGB3 (0.45) GPR139ITGB1ITGB3ITGAVITGA2B
SCHEMBL7339636 0.85 GPR132 (0.50) GPR139GPR132ALDH1A1SMN1; SMN2KMT2A
SCHEMBL7823171 0.83 ITGB3 (0.50) ITGB1ITGB3ITGAVITGA2BITGB5
SCHEMBL7340682 0.83 ALDH1A1 (0.47) GPR139ITGB1ITGB3ITGAVITGA2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0850221-B1 META-GUANIDINE, UREA, THIOUREA OR AZACYCLIC AMINO BENZOIC ACID DERIVATIVES AS INTEGRIN ANTAGONISTS SEARLE & CO (US) 2001-07-18 EP claimed