SCHEMBL7834591

SCHEMBL7834591

c1ccc2c(c1)CCCC2CSc1ncnc2nc[nH]c12

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CDC7 O00311 11/20 0.50
DBF4 Q9UBU7 11/20 0.50
RAB9A P51151 3/20 0.49
LMNA P02545 3/20 0.49
HTT P42858 3/20 0.49
NPC1 O15118 2/20 0.49
TSHR P16473 1/20 0.46
CYP1A2 P05177 3/20 0.46
SMN1; SMN2 Q16637 2/20 0.46
ALDH1A1 P00352 2/20 0.46
HPGD P15428 2/20 0.46
HIF1A Q16665 1/20 0.46
HTR3E A5X5Y0 1/20 0.45
MEN1 O00255 1/20 0.45
HTR3B O95264 1/20 0.45
MAPT P10636 1/20 0.45
HTR3A P46098 1/20 0.45
KMT2A Q03164 1/20 0.45
HTR3C Q8WXA8 1/20 0.45
CYP3A4 P08684 2/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7830640 0.81 G6PD (0.46) CDC7DBF4RAB9ALMNAHTT
SCHEMBL7835862 0.81 LMNA (0.41) CDC7DBF4LMNAHTTTSHR
SCHEMBL7834428 0.79 CYP19A1 (0.39) RAB9ANPC1KDM4E
SCHEMBL7830573 0.79 CDK1 (0.56) CDC7DBF4LMNAHTTTSHR
SCHEMBL7834228 0.71 CDK1 (0.46) CDC7DBF4LMNAHTTTSHR
SCHEMBL7821333 0.69 HTR6 (0.41)
Hydrochloric Acid SCHEMBL7822348 0.68 HTR6 (0.41) ALDH1A1MEN1KMT2ACYP2D6
SCHEMBL8808559 0.68 CYP19A1 (0.49) SMN1; SMN2ALDH1A1CYP2D6
SCHEMBL7822183 0.68 CDC7 (0.62) CDC7DBF4LMNAHTTCYP1A2
SCHEMBL29851680 0.68 CDC7 (1.00) CDC7DBF4RAB9ALMNAHTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0802914-B1 ARYL- AND HETEROARYL- PURINE AND PYRIDOPYRIMIDINE DERIVATIVES PHARMACIA & UPJOHN SPA (IT) 2001-06-06 EP claimed
EP-0802914-A1 ARYL AND HETEROARYL PURINE COMPOUNDS PHARMACIA & UPJOHN S.p.A. (IT) 1997-10-29 EP claimed
WO-1997018212-A1 ARYL AND HETEROARYL PURINE COMPOUNDS PHARMACIA & UPJOHN S.P.A. (IT) 1997-05-22 WO claimed
EP-0802914-B1 ARYL- AND HETEROARYL- PURINE AND PYRIDOPYRIMIDINE DERIVATIVES PHARMACIA & UPJOHN SPA (IT) 2001-06-06 EP disclosed
US-5965563-A NOVEL PURINE DERIVATIVES SUCH AS N6-(2-OXINDOL-5-YL) ADENINE, METHODS OF SYNTHESIZING THEM; USE AS TYROSINE KINASE INHIBITORS PHARMACIA & UPJOHN S.P.A. (IT) 1999-10-12 US disclosed