SCHEMBL7835862

SCHEMBL7835862

c1ccc2c(c1)CCCC2Cc1ncnc2nc[nH]c12

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LMNA P02545 6/20 0.41
HSD17B10 Q99714 3/20 0.41
TSHR P16473 2/20 0.41
HTT P42858 4/20 0.39
PKM P14618 2/20 0.39
CLK1 P49759 1/20 0.39
ADRA2A P08913 1/20 0.39
ADRA1D P25100 1/20 0.39
ADRA1A P35348 1/20 0.39
ADRA1B P35368 1/20 0.39
HTR6 P50406 1/20 0.39
CDK2 P24941 2/20 0.38
CDK1 P06493 1/20 0.38
CYP19A1 P11511 1/20 0.38
TBXAS1 P24557 1/20 0.38
PAK1 Q13153 1/20 0.38
CDC7 O00311 2/20 0.37
DBF4 Q9UBU7 2/20 0.37
AKT2 P31751 1/20 0.37
METAP2 P50579 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7830573 0.81 CDK1 (0.56) LMNAHSD17B10TSHRHTTPKM
SCHEMBL7834591 0.81 CDC7 (0.50) LMNAHSD17B10TSHRHTTPKM
SCHEMBL7822155 0.79 LMNA (0.40) LMNAHSD17B10TSHRHTTPKM
SCHEMBL7834141 0.77 CYP19A1 (0.41) ADRA2AADRA1DADRA1AADRA1BHTR6
SCHEMBL7821333 0.76 HTR6 (0.41) CLK1ADRA2AADRA1DADRA1AADRA1B
Hydrochloric Acid SCHEMBL7822348 0.75 HTR6 (0.41) CLK1ADRA2AADRA1DADRA1AADRA1B
SCHEMBL7830640 0.75 G6PD (0.46) LMNAHSD17B10TSHRHTTPKM
SCHEMBL7834228 0.74 CDK1 (0.46) LMNAHSD17B10TSHRHTTPKM
SCHEMBL7836198 0.72 SIGMAR1 (0.39) HTR6CYP19A1TBXAS1
Sulfuric Acid SCHEMBL7832166 0.70 HTR6 (0.40) HTR6CYP19A1TBXAS1CYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0802914-B1 ARYL- AND HETEROARYL- PURINE AND PYRIDOPYRIMIDINE DERIVATIVES PHARMACIA & UPJOHN SPA (IT) 2001-06-06 EP claimed
EP-0802914-A1 ARYL AND HETEROARYL PURINE COMPOUNDS PHARMACIA & UPJOHN S.p.A. (IT) 1997-10-29 EP claimed
WO-1997018212-A1 ARYL AND HETEROARYL PURINE COMPOUNDS PHARMACIA & UPJOHN S.P.A. (IT) 1997-05-22 WO claimed
EP-0802914-B1 ARYL- AND HETEROARYL- PURINE AND PYRIDOPYRIMIDINE DERIVATIVES PHARMACIA & UPJOHN SPA (IT) 2001-06-06 EP disclosed
US-5965563-A NOVEL PURINE DERIVATIVES SUCH AS N6-(2-OXINDOL-5-YL) ADENINE, METHODS OF SYNTHESIZING THEM; USE AS TYROSINE KINASE INHIBITORS PHARMACIA & UPJOHN S.P.A. (IT) 1999-10-12 US disclosed
EP-0802914-A1 ARYL AND HETEROARYL PURINE COMPOUNDS PHARMACIA & UPJOHN S.p.A. (IT) 1997-10-29 EP disclosed
WO-1997018212-A1 ARYL AND HETEROARYL PURINE COMPOUNDS PHARMACIA & UPJOHN S.P.A. (IT) 1997-05-22 WO disclosed