SCHEMBL7838799

SCHEMBL7838799

O=C(NC(CO)COc1ccccc1)c1c[nH]cn1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MTNR1A P48039 3/20 0.41
MTNR1B P49286 3/20 0.41
ADRB1 P08588 2/20 0.37
ADRB3 P13945 2/20 0.37
MMP2 P08253 2/20 0.37
MMP9 P14780 2/20 0.37
MMP12 P39900 2/20 0.37
PPARG P37231 1/20 0.36
PPARA Q07869 1/20 0.36
GPR88 Q9GZN0 1/20 0.36
F10 P00742 2/20 0.35
MME P08473 2/20 0.35
HDAC3 O15379 1/20 0.35
HDAC4 P56524 1/20 0.35
HDAC1 Q13547 1/20 0.35
HDAC7 Q8WUI4 1/20 0.35
HDAC2 Q92769 1/20 0.35
HDAC10 Q969S8 1/20 0.35
HDAC11 Q96DB2 1/20 0.35
HDAC8 Q9BY41 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7453033 0.80 CTSG (0.44) MMELMNAROCK2RPS6KA5RPS6KA4
SCHEMBL7836204 0.76 ROCK2 (0.50) ROCK2RPS6KA5PRKACAMAPK1GSK3A
SCHEMBL19357562 0.76 MTNR1A (0.53) MTNR1AMTNR1BADRB1ADRB3PPARG
SCHEMBL17104375 0.73 AKR1B1 (0.46) MME
SCHEMBL17104373 0.73 AKR1B1 (0.46) MME
SCHEMBL9089182 0.73 ALDH1A1 (0.55) MAPK1
SCHEMBL7827408 0.71 CNR1 (0.47)
SCHEMBL7835522 0.71 PDE5A (0.38) MMEHDAC6ROCK2ROCK1
SCHEMBL3008343 0.70 SMN1; SMN2 (0.41)
SCHEMBL7453024 0.70 MMP13 (0.40)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1098885-A1 IMIDAZOLE COMPOUNDS AND THEIR USE AS ADENOSINE DEAMINASE INHIBITORS FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 2001-05-16 EP disclosed
WO-2000005217-A1 IMIDAZOLE COMPOUNDS AND THEIR USE AS ADENOSINE DEAMINASE INHIBITORS FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 2000-02-03 WO disclosed