SCHEMBL7840730

SCHEMBL7840730

NC(=O)c1cccc(CCC(CO)NC(=O)c2c[nH]cn2)c1

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CTSG P08311 1/20 0.36
CTRB1 P17538 1/20 0.36
F10 P00742 3/20 0.36
F2 P00734 2/20 0.36
PRSS1 P07477 1/20 0.36
PRSS2 P07478 1/20 0.36
PRSS3 P35030 1/20 0.36
FOLH1 Q04609 1/20 0.35
ENPP2 Q13822 1/20 0.35
MEP1B Q16820 1/20 0.34
VNN1 O95497 1/20 0.34
ADA P00813 2/20 0.34
AURKA O14965 2/20 0.34
RPS6KB1 P23443 2/20 0.34
AURKB Q96GD4 2/20 0.34
KDM1A O60341 1/20 0.34
MAOA P21397 1/20 0.34
MAOB P27338 1/20 0.34
F3 P13726 1/20 0.34
CDC7 O00311 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7835522 0.86 PDE5A (0.38) CTSGCTRB1ROCK2EGFRROCK1
SCHEMBL7457472 0.85 CYP4F2 (0.48) MEP1BDYRK3CDK2CDK5DYRK1A
SCHEMBL7453024 0.85 MMP13 (0.40) EGFRCNR1PDE5A
SCHEMBL7453033 0.84 CTSG (0.44) CTSGCTRB1ADAROCK2RPS6KA5
SCHEMBL7840061 0.82 TAS1R3 (0.42) EGFRCNR1
SCHEMBL7452027 0.82 PDE5A (0.41) CTSGCTRB1F10F2ROCK2
SCHEMBL7827408 0.78 CNR1 (0.47) CNR1
SCHEMBL27521385 0.74 ADA (0.39) CTSGCTRB1ADAMAPK1GSK3B
SCHEMBL3649580 0.69 F3 (0.49) F3
SCHEMBL7838799 0.69 MTNR1A (0.41) F10ROCK2RPS6KA5MAPK1GSK3A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1098885-A1 IMIDAZOLE COMPOUNDS AND THEIR USE AS ADENOSINE DEAMINASE INHIBITORS FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 2001-05-16 EP disclosed
WO-2000005217-A1 IMIDAZOLE COMPOUNDS AND THEIR USE AS ADENOSINE DEAMINASE INHIBITORS FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 2000-02-03 WO disclosed