SCHEMBL7842740

SCHEMBL7842740

O=C(O)C(=O)c1cc(O)c(Cl)cc1F

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HPGD P15428 3/20 0.38
TSHR P16473 2/20 0.38
HSD17B10 Q99714 1/20 0.38
PYGL P06737 1/20 0.35
CES2 O00748 2/20 0.35
CES1 P23141 2/20 0.35
KEAP1 Q14145 1/20 0.35
NFE2L2 Q16236 1/20 0.35
HSP90AA1 P07900 3/20 0.35
POLB P06746 1/20 0.35
APEX1 P27695 1/20 0.35
CA2 P00918 2/20 0.34
HSD17B1 P14061 1/20 0.34
HSD17B2 P37059 1/20 0.34
PIK3CA P42336 1/20 0.33
MAPT P10636 1/20 0.33
CA1 P00915 1/20 0.33
AKR1C4 P17516 1/20 0.33
AKR1C3 P42330 1/20 0.33
AKR1C2 P52895 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7069337 0.84 KEAP1 (0.46) HPGDTSHRHSD17B10PYGLKEAP1
SCHEMBL6284961 0.79 RAB9A (0.46) HPGDPYGLPOLBMAPTALDH1A1
SCHEMBL9618645 0.78 HSP90AA1 (0.40) HPGDTSHRHSD17B10HSP90AA1POLB
SCHEMBL18013115 0.76 KEAP1 (0.46) HPGDTSHRHSD17B10PYGLKEAP1
SCHEMBL30471619 0.74 CES2 (0.43) HPGDCES2CES1KEAP1NFE2L2
SCHEMBL21239984 0.74 CES2 (0.43) HPGDCES2CES1KEAP1NFE2L2
SCHEMBL9617792 0.74 CA12 (0.44) HPGDTSHRPOLBAPEX1CA2
SCHEMBL23706639 0.72 PYGL (0.50) HPGDTSHRHSD17B10PYGLKEAP1
SCHEMBL18893969 0.71 HSD17B10 (0.55) HPGDTSHRHSD17B10HSP90AA1POLB
SCHEMBL7840274 0.71 CES2 (0.50) TSHRCES2CES1CA2CA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1306523-A Substituted 6-aryl-3-thioxo-5-(thi) oxo-2,3,4,5-tetrahydro-1,2,4-triazines BASF AG (DE) 2001-08-01 CN disclosed
EP-1077954-A1 SUBSTITUTED 6-ARYL-3-THIOXO-5-(THI)OXO-2,3,4,5-TETRAHYDRO-1,2,4-TRIAZINES BASF AKTIENGESELLSCHAFT (DE) 2001-02-28 EP disclosed
WO-1999059983-A1 SUBSTITUTED 6-ARYL-3-THIOXO-5-(THI)OXO-2,3,4,5-TETRAHYDRO-1,2,4-TRIAZINES BASF AKTIENGESELLSCHAFT (DE) 1999-11-25 WO disclosed