SCHEMBL7844303

SCHEMBL7844303

NC(=O)c1ccc(F)c(C(N)=O)c1Cc1ccc(F)cc1

nearest known ligand 0.43

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
MAPK8 P45983 2/20 0.40
MAOB P27338 2/20 0.38
PARP10 Q53GL7 1/20 0.38
RPS6KB1 P23443 3/20 0.38
DGAT1 O75907 1/20 0.37
PARP1 P09874 3/20 0.36
ALDH1A1 P00352 1/20 0.35
TAAR1 Q96RJ0 1/20 0.35
AKT1 P31749 1/20 0.35
LMNA P02545 1/20 0.35
HTT P42858 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.35
AGTR1 P30556 1/20 0.35
AURKA O14965 1/20 0.34
IDO1 P14902 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28349448 0.82 PSIP1 (0.42) PARP1ALDH1A1
SCHEMBL27895663 0.80 RPS6KB1 (0.46) MAPK8MAOBPARP10RPS6KB1PARP1
SCHEMBL184570 0.80 MAPK8 (0.39) MAPK8MAOBPARP10RPS6KB1ALDH1A1
SCHEMBL28974830 0.76 MAPT (0.40) MAPK8MAOBPARP10RPS6KB1ALDH1A1
SCHEMBL28128227 0.75 LMNA (0.44) MAPK8MAOBDGAT1ALDH1A1LMNA
SCHEMBL28127954 0.75 DGAT1 (0.51) MAPK8PARP10RPS6KB1DGAT1PARP1
SCHEMBL28658004 0.75 RPS6KB1 (0.42) MAPK8MAOBPARP10RPS6KB1PARP1
SCHEMBL27970605 0.74 MAPK8 (0.39) MAPK8MAOBPARP10RPS6KB1ALDH1A1
SCHEMBL9018997 0.72 KMT2A (0.39) DGAT1PARP1ALDH1A1LMNA
SCHEMBL1990289 0.71 CYP3A4 (0.50) PARP10RPS6KB1ALDH1A1AURKA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1150565-A1 THIAZOLE DERIVATIVES AND COMBINATORIAL LIBRARIES THEREOF LION bioscience AG (DE) 2001-11-07 EP claimed
WO-2000045635-A1 THIAZOLE DERIVATIVES AND COMBINATORIAL LIBRARIES THEREOF LION BIOSCIENCE AG (DE) 2000-08-10 WO claimed