SCHEMBL7844409

SCHEMBL7844409

c1ccc(COc2ccc3cc(OCc4cn(C(c5ccccc5)(c5ccccc5)c5ccccc5)cn4)ccc3c2)cc1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALOX5 P09917 2/20 0.52
CYP3A4 P08684 2/20 0.45
NPC1 O15118 3/20 0.43
RAB9A P51151 2/20 0.43
MEN1 O00255 2/20 0.42
KMT2A Q03164 2/20 0.42
MRGPRX4 Q96LA9 1/20 0.42
ACSS2 Q9NR19 1/20 0.42
ROCK1 Q13464 1/20 0.41
SIRT2 Q8IXJ6 6/20 0.41
CA12 O43570 1/20 0.40
CA1 P00915 1/20 0.40
CA2 P00918 1/20 0.40
CA3 P07451 1/20 0.40
MAOA P21397 1/20 0.40
CA4 P22748 1/20 0.40
CA6 P23280 1/20 0.40
MAOB P27338 1/20 0.40
CA7 P43166 1/20 0.40
MTNR1A P48039 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7818117 0.89 SIRT2 (0.44) NPC1RAB9ASIRT2MAOB
SCHEMBL224236 0.84 SIRT2 (0.43) SIRT2
SCHEMBL7594682 0.84 SIRT2 (0.41) NPC1RAB9ASIRT2CA12CA1
SCHEMBL6674214 0.84 KCNH2 (0.46) SIRT2
SCHEMBL7597443 0.81 MAOA (0.39) MRGPRX4SIRT2CA12MAOAMAOB
SCHEMBL5203299 0.80 MAOB (0.50) CYP3A4SIRT2MAOB
SCHEMBL5751662 0.80 ALOX5 (0.44) ALOX5CYP3A4NPC1RAB9AMEN1
SCHEMBL5750032 0.80 ALOX5 (0.44) ALOX5NPC1MEN1KMT2AMRGPRX4
SCHEMBL7384162 0.79 ALDH1A1 (0.53) RAB9AMEN1KMT2ASIRT2
SCHEMBL5747790 0.78 ALOX5 (0.45) ALOX5CYP3A4NPC1RAB9AMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1073640-A1 NAPHTHALENE DERIVATIVES, THEIR PRODUCTION AND USE Takeda Chemical Industries, Ltd. (JP) 2001-02-07 EP disclosed
WO-1999054309-A1 NAPHTHALENE DERIVATIVES, THEIR PRODUCTION AND USE TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1999-10-28 WO disclosed