SCHEMBL7597443

SCHEMBL7597443

c1ccc(C(c2ccccc2)(c2ccccc2)n2cnc(COc3ccc4c(ccc5occc54)c3)c2)cc1

nearest known ligand 0.40

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
MAOA P21397 4/20 0.39
MAOB P27338 4/20 0.39
MRGPRX4 Q96LA9 2/20 0.36
KCNA3 P22001 2/20 0.36
KCNA5 P22460 1/20 0.36
SIRT2 Q8IXJ6 8/20 0.36
CA12 O43570 2/20 0.34
CA9 Q16790 2/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7844409 0.81 ALOX5 (0.52) MAOAMAOBMRGPRX4SIRT2CA12
SCHEMBL7818117 0.80 SIRT2 (0.44) MAOBSIRT2
SCHEMBL7594682 0.77 SIRT2 (0.41) SIRT2CA12CA9
SCHEMBL6674214 0.75 KCNH2 (0.46) SIRT2
SCHEMBL4027506 0.75 ENPP2 (0.31) SIRT2
SCHEMBL7828102 0.74 SIRT2 (0.40) SIRT2
SCHEMBL4031880 0.74 CTNNB1 (0.34) SIRT2
SCHEMBL7831405 0.72 SIRT2 (0.35) SIRT2
SCHEMBL5203299 0.72 MAOB (0.50) MAOBSIRT2
SCHEMBL7384162 0.70 ALDH1A1 (0.53) SIRT2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1222174-A1 IMIDAZOL-4-YLMETHANOLS USED AS INHIBITORS OF STEROID C17-20 LYASE Takeda Chemical Industries, Ltd. (JP) 2002-07-17 EP disclosed
WO-2001030762-A1 IMIDAZOL-4-YLMETHANOLS USE AS INHIBITORS OF STEROID C17-20 LYASE TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 2001-05-03 WO disclosed