SCHEMBL7849232

SCHEMBL7849232

CC(C)C[C@@H](CNN1C(=O)NC2(CCN(C(=O)OCc3ccccc3)CC2)C1=O)[C@H](CCCc1ccccc1)C(=O)NO

nearest known ligand 0.40

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
HDAC1 Q13547 3/20 0.40
HDAC6 Q9UBN7 3/20 0.40
HDAC3 O15379 2/20 0.40
HDAC2 Q92769 2/20 0.40
SCN5A Q14524 1/20 0.37
SCN9A Q15858 1/20 0.37
XIAP P98170 1/20 0.35
BIRC2 Q13490 1/20 0.35
CTSK P43235 5/20 0.35
CTSL P07711 4/20 0.35
CTSS P25774 3/20 0.35
MMP8 P22894 1/20 0.35
MMP2 P08253 1/20 0.35
MMP9 P14780 1/20 0.35
ADAM17 P78536 1/20 0.35
CTSB P07858 2/20 0.35
HDAC8 Q9BY41 1/20 0.34
MMP1 P03956 1/20 0.34
MMP13 P45452 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7848203 0.89 L3MBTL1 (0.35) SCN5ASCN9ACTSKCTSLCTSS
SCHEMBL7849143 0.88 HDAC1 (0.41) HDAC1HDAC6HDAC3HDAC2SCN5A
SCHEMBL7955667 0.82 MMP1 (0.40) MMP8MMP2MMP9ADAM17MMP1
SCHEMBL7836622 0.82 SIGMAR1 (0.34) MMP9MMP1
SCHEMBL7955182 0.80 MEN1 (0.39) HDAC1HDAC6HDAC3HDAC2SCN5A
SCHEMBL7848201 0.77 L3MBTL1 (0.36) SCN5ASCN9ACTSKCTSLCTSS
SCHEMBL7946527 0.75 MMP1 (0.43) MMP8MMP2MMP9ADAM17MMP1
SCHEMBL7946524 0.75 MMP1 (0.43) MMP8MMP2MMP9ADAM17MMP1
SCHEMBL7955660 0.74 XIAP (0.35) XIAPBIRC2CTSKCTSLCTSS
SCHEMBL7955777 0.74 MMP1 (0.45) MMP8MMP2MMP9ADAM17MMP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1137640-A1 CYCLIC HYDRAZINE DERIVATIVES AS TNF-ALPHA INHIBITORS F. HOFFMANN-LA ROCHE AG (CH) 2001-10-04 EP disclosed
WO-2000035885-A1 CYCLIC HYDRAZINE DERIVATIVES AS TNF-ALPHA INHIBITORS F. HOFFMANN-LA ROCHE AG (CH) 2000-06-22 WO disclosed