SCHEMBL7852248

SCHEMBL7852248

CC(C)(C)OC(=O)N(C(=O)[C@@H](N)CC(=O)O)[C@@H](CC1CCCCC1)C(=O)OC(c1ccccc1)c1ccccc1

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MMP1 P03956 5/20 0.37
MMP2 P08253 5/20 0.37
MMP3 P08254 5/20 0.37
REN P00797 3/20 0.36
KIF11 P52732 1/20 0.35
METAP2 P50579 2/20 0.34
METAP1 P53582 2/20 0.34
CTSL P07711 1/20 0.34
CTSB P07858 1/20 0.34
CTSS P25774 1/20 0.34
CTSK P43235 1/20 0.34
PSEN1 P49768 3/20 0.34
PSEN2 P49810 3/20 0.34
APH1B Q8WW43 3/20 0.34
NCSTN Q92542 3/20 0.34
APH1A Q96BI3 3/20 0.34
PSENEN Q9NZ42 3/20 0.34
HTR2C P28335 2/20 0.33
SLC6A4 P31645 2/20 0.33
OPRK1 P41145 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7207592 0.78 CTSL (0.40) MMP1MMP2MMP3RENCTSL
SCHEMBL7204995 0.74 MMP2 (0.50) MMP1MMP2MMP3METAP2METAP1
SCHEMBL15259739 0.73 CHRNB2 (0.36) KIF11CTSSCTSK
Hydrochloric Acid SCHEMBL7205141 0.73 MMP2 (0.49) MMP1MMP2MMP3METAP2METAP1
SCHEMBL7852251 0.73 FAAH (0.39) MMP1MMP2MMP3CTSLCTSB
SCHEMBL7852245 0.72 CTSS (0.52) MMP1MMP2MMP3RENCTSS
SCHEMBL7205030 0.71 MMP2 (0.48) MMP1MMP2MMP3KIF11METAP2
SCHEMBL7210238 0.71 OPRK1 (0.36) MMP1MMP2MMP3RENMETAP2
SCHEMBL7212756 0.70 KLK7 (0.36) MMP1MMP2MMP3RENMETAP2
SCHEMBL7852252 0.70 OPRK1 (0.36) MMP1MMP2MMP3RENMETAP2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6180759-B1 PREPARING AZACYCLOALKANOYLPSEUDOTETRAPEPTIDES COMPRISING COUPLING A DIPEPTIDE WITH A PSEUDODIPEPTIDE; FOR EXAMPLE, N-(N-ETHYL-N-(1-OXO-4-(4-PIPERIDINYL)BUTYL)GLYCYL)-(L)-ALPHA-ASPARTYL-3 -CYCLOHEXYL-(L)-ALANINEAMIDE; USE AS ANTICOAGULANTS AVENTIS PHARMACEUTICALS PRODUCTS INC. 2001-01-30 US disclosed