SCHEMBL7860078

SCHEMBL7860078

CCOC(=O)C(Cc1ccccc1)(Oc1ccccc1OCCc1ccccc1)C(=O)OCC

nearest known ligand 0.47

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.47
RECQL P46063 1/20 0.47
MMP8 P22894 1/20 0.47
ABCB1 P08183 1/20 0.43
PPARG P37231 4/20 0.41
PTGES O14684 3/20 0.41
ALOX5 P09917 3/20 0.41
TAAR1 Q96RJ0 2/20 0.40
THRB P10828 1/20 0.40
PIN1 Q13526 1/20 0.40
KMT2A Q03164 1/20 0.39
PPID Q08752 1/20 0.39
GLA P06280 1/20 0.39
L3MBTL1 Q9Y468 1/20 0.39
PPARD Q03181 1/20 0.39
PPARA Q07869 1/20 0.39
FFAR1 O14842 1/20 0.39
MAPT P10636 1/20 0.39
SMN1; SMN2 Q16637 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7861235 0.88 ALDH1A1 (0.48) ALDH1A1RECQLMMP8L3MBTL1MAPT
SCHEMBL9206341 0.85 KMT2A (0.48) ALDH1A1RECQLMMP8KMT2AGLA
SCHEMBL9199837 0.82 ALDH1A1 (0.47) ALDH1A1RECQLMMP8PIN1PPID
SCHEMBL16865453 0.76 ALDH1A1 (0.57) ALDH1A1RECQLMMP8TAAR1THRB
SCHEMBL7431853 0.76 ALDH1A1 (0.57) ALDH1A1RECQLMMP8ABCB1TAAR1
SCHEMBL7860005 0.75 ABCB1 (0.51) ABCB1KMT2AGLAL3MBTL1FFAR1
SCHEMBL7854590 0.75 TDP1 (0.47) ALDH1A1MMP8ABCB1PPARGPTGES
SCHEMBL7854387 0.74 ALDH1A1 (0.45) ALDH1A1L3MBTL1MAPT
SCHEMBL7861112 0.74 ATM (0.45) ALDH1A1KMT2AL3MBTL1MAPT
SCHEMBL20350605 0.74 MMP8 (0.58) ALDH1A1RECQLMMP8TAAR1THRB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0625969-B1 ARYLALKOXYPHENOXY-IMIDAZOLINE COMPOUNDS MERRELL PHARMA INC (US) 2001-03-07 EP disclosed
US-5407954-A Serotonin antagonism; treats depression, anxiety, hypertension and migraine headaches MERRELL DOW PHARMACEUTICALS INC. (US) 1995-04-18 US disclosed
EP-0625969-A1 ARYLALKOXYPHENOXY-IMIDAZOLINE COMPOUNDS MERRELL PHARMACEUTICALS INC. (US) 1994-11-30 EP disclosed
US-5216008-A Antidepressant, anxiolytic, hypotensive and also treats migraine headaches MERRELL DOW PHARMACEUTICALS INC. (US) 1993-06-01 US disclosed