SCHEMBL7860112

SCHEMBL7860112

CCC(CN1C=NCC1)c1ccccc1Oc1ccccc1OCc1ccc(N)cc1

nearest known ligand 0.31

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NISCH Q9Y2I1 1/20 0.31
RAB9A P51151 3/20 0.31
ALDH1A1 P00352 2/20 0.31
NPC1 O15118 2/20 0.31
HTR1A P08908 2/20 0.31
ADRA1D P25100 1/20 0.31
ADRA1A P35348 1/20 0.31
ADRA1B P35368 1/20 0.31
APP P05067 2/20 0.30
LTA4H P09960 1/20 0.30
MAPK14 Q16539 1/20 0.30
SMN1; SMN2 Q16637 2/20 0.30
GAA P10253 1/20 0.30
MAPT P10636 1/20 0.30
MAOA P21397 1/20 0.30
MAOB P27338 1/20 0.30
L3MBTL1 Q9Y468 1/20 0.30
KMT2A Q03164 1/20 0.30
SLC6A2 P23975 1/20 0.30
SLC6A4 P31645 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7861001 0.89 NPC1 (0.35) RAB9AALDH1A1NPC1HTR1AADRA1D
SCHEMBL7860121 0.89 NISCH (0.34) NISCHRAB9AALDH1A1NPC1HTR1A
SCHEMBL7861125 0.86 MEN1 (0.39) RAB9AALDH1A1NPC1HTR1AADRA1D
SCHEMBL7862260 0.80 CYP19A1 (0.34) RAB9AALDH1A1NPC1LTA4HMAPK14
SCHEMBL7860116 0.79 EZH2 (0.36) RAB9AALDH1A1NPC1HTR1AADRA1D
SCHEMBL7861310 0.78 MAPT (0.44) ALDH1A1HTR1AADRA1DADRA1AADRA1B
SCHEMBL7854338 0.77 HTR1A (0.36) RAB9AHTR1AAPPLTA4HMAPK14
SCHEMBL7864331 0.75 NPC1 (0.40) RAB9ANPC1HTR1AADRA1DADRA1A
SCHEMBL7861309 0.74 HTR6 (0.40) RAB9AALDH1A1NPC1MAPTL3MBTL1
SCHEMBL7859923 0.71 CYP19A1 (0.36) RAB9ANPC1HTR1ALTA4HMAPK14

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0625969-B1 ARYLALKOXYPHENOXY-IMIDAZOLINE COMPOUNDS MERRELL PHARMA INC (US) 2001-03-07 EP claimed
US-5407954-A Serotonin antagonism; treats depression, anxiety, hypertension and migraine headaches MERRELL DOW PHARMACEUTICALS INC. (US) 1995-04-18 US claimed
WO-1993016051-A1 ARYLALKOXYPHENOXY-IMIDAZOLINE COMPOUNDS MERRELL DOW PHARMACEUTICALS INC. (US) 1993-08-19 WO claimed
EP-0625969-B1 ARYLALKOXYPHENOXY-IMIDAZOLINE COMPOUNDS MERRELL PHARMA INC (US) 2001-03-07 EP disclosed
US-5407954-A Serotonin antagonism; treats depression, anxiety, hypertension and migraine headaches MERRELL DOW PHARMACEUTICALS INC. (US) 1995-04-18 US disclosed