SCHEMBL7860116

SCHEMBL7860116

CCC(CN1C=NCC1)c1ccc(Oc2ccccc2OCc2ccccc2)cc1

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
EZH2 Q15910 1/20 0.36
ALDH1A1 P00352 2/20 0.35
NPC1 O15118 2/20 0.34
ABCB1 P08183 1/20 0.34
KDM4E B2RXH2 1/20 0.34
MEN1 O00255 1/20 0.34
TP53 P04637 1/20 0.34
KMT2A Q03164 1/20 0.34
SMN1; SMN2 Q16637 1/20 0.34
NPSR1 Q6W5P4 1/20 0.34
FFAR1 O14842 1/20 0.34
LIPE Q05469 1/20 0.34
MAPT P10636 2/20 0.33
HRH3 Q9Y5N1 1/20 0.33
HTR1A P08908 1/20 0.33
ADRA1D P25100 1/20 0.33
ADRA1A P35348 1/20 0.33
ADRA1B P35368 1/20 0.33
GRIN1 Q05586 1/20 0.33
GRIN2B Q13224 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7861001 0.81 NPC1 (0.35) ALDH1A1NPC1HTR1AADRA1DADRA1A
SCHEMBL9445181 0.81 KDR (0.38) MAPTL3MBTL1
SCHEMBL7861310 0.77 MAPT (0.44) ALDH1A1KDM4EMEN1KMT2ASMN1; SMN2
SCHEMBL7861125 0.75 MEN1 (0.39) ALDH1A1NPC1MEN1KMT2ASMN1; SMN2
SCHEMBL7859944 0.72 HTR1A (0.41) ALDH1A1NPC1ABCB1KDM4EMEN1
SCHEMBL7862260 0.71 CYP19A1 (0.34) ALDH1A1NPC1LIPERAB9A
SCHEMBL7859937 0.71 LMNA (0.40) ALDH1A1KDM4EMEN1KMT2ANPSR1
SCHEMBL9252950 0.71 CHRNB2 (0.40) ALDH1A1NPC1KDM4EMEN1TP53
SCHEMBL7859925 0.70 HTR1A (0.46) ALDH1A1ABCB1KDM4EMEN1TP53
SCHEMBL7854567 0.70 MTNR1A (0.44) NPC1ABCB1HTR1ARAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0625969-B1 ARYLALKOXYPHENOXY-IMIDAZOLINE COMPOUNDS MERRELL PHARMA INC (US) 2001-03-07 EP claimed
WO-1993016051-A1 ARYLALKOXYPHENOXY-IMIDAZOLINE COMPOUNDS MERRELL DOW PHARMACEUTICALS INC. (US) 1993-08-19 WO claimed
US-5216008-A Antidepressant, anxiolytic, hypotensive and also treats migraine headaches MERRELL DOW PHARMACEUTICALS INC. (US) 1993-06-01 US claimed
EP-0625969-B1 ARYLALKOXYPHENOXY-IMIDAZOLINE COMPOUNDS MERRELL PHARMA INC (US) 2001-03-07 EP disclosed
US-5407954-A Serotonin antagonism; treats depression, anxiety, hypertension and migraine headaches MERRELL DOW PHARMACEUTICALS INC. (US) 1995-04-18 US disclosed
US-5216008-A Antidepressant, anxiolytic, hypotensive and also treats migraine headaches MERRELL DOW PHARMACEUTICALS INC. (US) 1993-06-01 US disclosed