SCHEMBL7861944

SCHEMBL7861944

N=C(N)Nc1cccc(/C=C/c2cccc(C(CC(=O)O)c3ccccc3)c2)c1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HDAC1 Q13547 1/20 0.45
SNCA P37840 2/20 0.42
PKM P14618 1/20 0.41
HDAC4 P56524 1/20 0.40
MEF2D Q14814 1/20 0.40
MAPT P10636 2/20 0.39
POLB P06746 1/20 0.39
MAPK1 P28482 1/20 0.39
CYP2C19 P33261 2/20 0.38
ALDH1A1 P00352 2/20 0.38
SIRT1 Q96EB6 1/20 0.38
MEN1 O00255 1/20 0.38
LMNA P02545 1/20 0.38
CYP1A2 P05177 1/20 0.38
KMT2A Q03164 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.38
TDP1 Q9NUW8 1/20 0.38
ITGB3 P05106 2/20 0.38
ITGA2B P08514 2/20 0.38
PARP1 P09874 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7856431 1.00 HDAC1 (0.45) HDAC1SNCAPKMHDAC4MEF2D
SCHEMBL7863285 0.82 ITGB3 (0.48) MAPTPOLBMAPK1ALDH1A1SIRT1
SCHEMBL7864754 0.81 PTPN11 (0.48) MAPTPOLBMAPK1ALDH1A1LMNA
SCHEMBL7856433 0.81 ITGB3 (0.54) MAPTPOLBMEN1KMT2ASMN1; SMN2
SCHEMBL7856428 0.80 PARP1 (0.44) PKMMAPTPOLBMAPK1ALDH1A1
SCHEMBL7863273 0.79 FFAR1 (0.43) HDAC4MEF2DMAPTPOLBMAPK1
SCHEMBL7455765 0.78 ITGB3 (0.58) HDAC1POLBALDH1A1SIRT1MEN1
SCHEMBL7862046 0.77 ITGB3 (0.45) PKMMAPTPOLBMEN1KMT2A
SCHEMBL7863151 0.77 KMT2A (0.57) SIRT1MEN1KMT2ASMN1; SMN2
SCHEMBL7864761 0.77 ITGB3 (0.43) MAPTPOLBCYP2C19MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0889877-B1 META-SUBSTITUTED PHENYLENE DERIVATIVES AND THEIR USE AS ALPHAvBETA3 INTEGRIN ANTAGONISTS OR INHIBITORS SEARLE & CO (US) 2001-08-29 EP claimed
EP-0889877-B1 META-SUBSTITUTED PHENYLENE DERIVATIVES AND THEIR USE AS ALPHAvBETA3 INTEGRIN ANTAGONISTS OR INHIBITORS SEARLE & CO (US) 2001-08-29 EP disclosed