SCHEMBL7861972

SCHEMBL7861972

CC(C)(C)OC(=O)CC(c1ccccc1)c1cccc(NS(=O)(=O)c2cccc(NC(N)=S)c2)c1

nearest known ligand 0.43

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
TGFBR1 P36897 2/20 0.43
MEN1 O00255 3/20 0.41
KMT2A Q03164 3/20 0.41
F2 P00734 3/20 0.41
MAPT P10636 5/20 0.40
LMNA P02545 2/20 0.40
ALDH1A1 P00352 1/20 0.40
PKM P14618 1/20 0.40
MAPK1 P28482 1/20 0.40
CASR P41180 1/20 0.40
IDH1 O75874 2/20 0.39
F10 P00742 1/20 0.39
PRSS1 P07477 1/20 0.39
CA1 P00915 2/20 0.39
CA2 P00918 2/20 0.39
GAA P10253 1/20 0.39
TMPRSS6 Q8IU80 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7861844 0.93 CA1 (0.47) TGFBR1MEN1KMT2AF2MAPT
SCHEMBL7863291 0.86 ITGB3 (0.45) MEN1KMT2AMAPTPKMCA1
SCHEMBL7856493 0.85 NAMPT (0.53) MEN1KMT2AMAPTLMNAMAPK1
SCHEMBL7864640 0.81 TGFBR1 (0.39) TGFBR1MEN1KMT2AF2MAPT
SCHEMBL7861968 0.81 TGFBR1 (0.39) TGFBR1MEN1KMT2AF2MAPT
SCHEMBL7861976 0.81 CA12 (0.43) TGFBR1MEN1KMT2AMAPTLMNA
SCHEMBL7856530 0.78 CA1 (0.54) MEN1KMT2AMAPTPKMCA1
SCHEMBL7862046 0.76 ITGB3 (0.45) MEN1KMT2AF2MAPTPKM
SCHEMBL7856438 0.75 CASR (0.49) MEN1KMT2AMAPTCASR
SCHEMBL7863294 0.74 HTR6 (0.48) MEN1KMT2AMAPTLMNAALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0889877-B1 META-SUBSTITUTED PHENYLENE DERIVATIVES AND THEIR USE AS ALPHAvBETA3 INTEGRIN ANTAGONISTS OR INHIBITORS SEARLE & CO (US) 2001-08-29 EP claimed
EP-0889877-B1 META-SUBSTITUTED PHENYLENE DERIVATIVES AND THEIR USE AS ALPHAvBETA3 INTEGRIN ANTAGONISTS OR INHIBITORS SEARLE & CO (US) 2001-08-29 EP disclosed
US-5773646-A INTEGRIN INHIBITORS G. D. SEARLE & CO. (US) 1998-06-30 US disclosed